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3-({ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-N-(1-methyl-1H-pyrazol-4-yl)benzamide
5-{1-[(2-chlorophenyl)methyl]-1H-imidazol-2-yl}-2-(pyridin-2-yl)pyrimidine
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-4-(1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
8-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2E)-N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
3-{2-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
2,6-dimethyl-N-[2-(pyridin-3-yloxy)propyl]quinoline-4-carboxamide
ethyl 2-[1-(5-chloro-2-hydroxybenzoyl)piperidin-2-yl]acetate
methyl 1-({4-[3-(pyridin-2-yl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
thiophen-2-yl(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)methanol
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-(pyridin-2-yl)acetamide
2-{4-[2-(propan-2-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
(4aS,8aR)-2-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-decahydroisoquinoline
3-chloro-4-[(1-cyclohexylpiperidin-4-yl)oxy]-N-cyclopentylbenzamide
3-(4H-1,2,4-triazol-4-yl)adamantan-1-ol
3-cyano-N-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
2-methoxy-N-(3-methyl-1-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
1-methyl-N-{[2-(trifluoromethoxy)phenyl]methyl}piperidine-2-carboxamide
5-[4-(1H-pyrrole-2-carbonyl)piperazine-1-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(thiophen-2-ylmethyl)acetamide
(2S,4R)-N-ethyl-1-[(2-fluorophenyl)methyl]-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
3-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-(2-fluoro-4-methylphenyl)urea
N-[2-(2,4-difluorophenyl)-1-{1-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]piperidin-4-yl}ethyl]-N-methylpropanamide
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-3-hydroxypropan-1-one
5-benzenesulfonamido-1-ethyl-2-methyl-N-(oxolan-3-yl)-1H-1,3-benzodiazole-7-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}propanamide
N-(3-ethoxypropyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
1-{1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-4-yl}pyrrolidin-2-one
1-ethyl-3-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
4-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-2,6-dimethylpyrimidine
2-(furan-2-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-oxoacetamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-[(2R,3R)-1'-(5-acetylthiophene-3-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
3-[(3,4-dimethylphenyl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(3-hydroxypropyl)-1-(3-methanesulfonamidophenyl)-3-(thiophen-2-ylmethyl)urea
N-[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-methyl-N-[2-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
N-butyl-2-[N-methyl-1-(2-methyl-1-benzofuran-5-yl)formamido]acetamide
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}){[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}amine
methyl(1,2-oxazol-3-ylmethyl){[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
1-[4-({[2-(dimethylamino)-6-ethylpyrimidin-4-yl]amino}methyl)piperidin-1-yl]-2-methylpropan-1-one
N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]pyridine-3-carboxamide
3-[2-(4-methanesulfonylphenyl)acetyl]-3,9-diazaspiro[5.6]dodecan-10-one
[(3R,5S)-5-(morpholin-4-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]methanol
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-ethyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
ethyl 1-{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}piperidine-3-carboxylate
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-phenylpropanamide
4-methoxy-N-(2-methoxyethyl)-2-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)oxy]benzamide