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2-cyclopropyl-N-methyl-6-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,6-dihydropyrimidine-5-carboxamide
methyl 1-(benzyloxy)-2-oxo-8-(quinolin-5-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
4-[6-(1-hydroxyethyl)pyridin-2-yl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-methyl-2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-1H-indole
N,N-diethyl-1-[(1s,4s)-4-propanamidocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
1-{1-[(4-fluoro-3-methoxyphenyl)methyl]azetidin-3-yl}piperidine
4-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}pyrimidin-2-amine
4-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyridine
3-[(3-ethoxyphenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
7-(3-chlorophenyl)-4-[(2-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-methyl-3-[(E)-2-phenylethenesulfonyl]-3,9-diazaspiro[5.6]dodecane
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}cyclopropanecarboxamide
N-[(1-benzylpiperidin-4-yl)methyl]pyrimidin-4-amine
N4-[(2,3-dimethyl-1H-indol-5-yl)methyl]-6-methylpyrimidine-2,4-diamine
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
(3S,4R)-3-benzyl-1-(2-methoxybenzenesulfonyl)-4-methylpiperidin-4-ol
(1R,5R)-3-benzoyl-6-(1H-indol-5-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]cyclohexane-1-carboxamide
N-[3-(ethylcarbamoyl)-5-[({[4-(trifluoromethoxy)phenyl]methyl}amino)methyl]phenyl]pyridine-2-carboxamide
2-methoxy-1-(4-{2-[2-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]bis(1,3-oxazol-4-ylmethyl)amine
1,3-dimethyl-5-[({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)methyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-{[2-(3-phenyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
(2S)-1-({1-[1-(2-methylpropanoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidine-2-carboxamide
6-[(4-ethylphenyl)methyl]-N-(2-methoxyphenyl)-6-azaspiro[2.5]octane-1-carboxamide
7-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-4-(piperidin-1-yl)butanamide
N-({8-[(4-ethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
2-amino-N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-{[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-(morpholin-4-yl)propyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]piperidin-2-one
3-(6-methoxyquinolin-8-yl)-1-[3-(morpholin-4-yl)propyl]urea
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-(1H-imidazol-2-ylmethyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
1-[2-(dimethylamino)ethyl]-N-(1H-imidazol-2-ylmethyl)-N-methyl-5-oxopyrrolidine-3-carboxamide
9-(6-aminopyridine-3-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(cyclohexylmethyl)-2-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[8-(2,6-dimethylquinoline-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
1-(4-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}piperidin-1-yl)-2-methylpropan-1-one
6-ethyl-2-oxo-N-(4-phenylbutyl)-1,2-dihydropyridine-4-carboxamide
3-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
N-[(3,5-dimethoxyphenyl)methyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
5-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
2-{[4-(pyrrolidine-1-sulfonyl)-1,4-diazepan-1-yl]methyl}benzonitrile
3-{1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]piperidin-3-yl}benzoic acid
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-{[3-methyl-7-(naphthalene-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-({1-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
3-{3-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]propoxy}pyridine