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1-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(2H-indazol-2-yl)ethan-1-one
1-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
(1R,3S)-3-(2-aminoethoxy)-7-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
2-amino-6-{4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperazin-1-yl}pyrimidin-4-ol
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-(2-methoxyphenyl)pyridazine
2-(2-methoxyethyl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-1,3-benzoxazole-6-carboxamide
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-6-(4-methoxyphenyl)-1,2-dihydropyridin-2-one
2-methyl-8-[(3-methyl-1,2-benzoxazol-5-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
ethyl 4-(4-{4-[(2-methylpropyl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
2-(2,4-difluorophenoxy)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}acetamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4,7-trimethyl-1H-indole-2-carboxamide
N,1-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
[9-(2-ethoxyethyl)-3-(2-methylpyridin-4-yl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
2-({4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-(1H-pyrazol-1-yl)propan-1-one
2-{[2-(2,3-dihydro-1H-isoindole-2-carbonyl)phenyl]amino}acetic acid
3-{[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]amino}-2-(thiophen-3-ylmethyl)propan-1-ol
4-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}phenol
ethyl 4-{[6-chloro-2-(dimethylcarbamoyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine-1-carboxylate
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
[(2,3-dimethoxyphenyl)methyl]({[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl})amine
3-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
5-chloro-N-(2-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)-3-methyl-1H-indole-2-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-propyl-1,3-thiazole-4-carboxamide
phenyl(1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-yl)methanol
N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-3-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
2-(2-fluoro-6-methoxyphenyl)-4-(pyrrolidine-1-carbonyl)pyridine
4-(pyrrolidin-1-ylmethyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-4-ol
1-(4-fluorophenyl)-3-methyl-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazole
2-(4-fluorophenyl)-N-{2-[7-(2-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
5-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-2,1,3-benzothiadiazole
5-(phenoxymethyl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
4-cyclopentyl-N-methyl-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
methyl (2S,4S,5R)-4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]carbamoyl}-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylate
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
3-acetyl-N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-1H-pyrazole-5-carboxamide
methyl 3-(oxolane-3-amido)-1-(2-phenylethyl)-5-[(1-propylpiperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-[1-(1H-pyrazol-3-ylmethyl)piperidin-4-yl]thiomorpholine
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
3-(2-amino-1,3-thiazol-4-yl)-1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]propan-1-one
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
N-(furan-2-ylmethyl)-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
N-cyclopentyl-1-[2-(dimethylamino)ethyl]-6-methyl-4-oxo-2-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[5-(oxan-2-yl)thiophen-2-yl]methyl}amine
N-(1-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
ethyl 5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-({4-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}methyl)-5-methylpyrazine