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(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)(thiophen-2-yl)methanol
2-(9-{[4-(methylsulfanyl)phenyl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetic acid
3-(2-methoxybenzoyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(methylsulfamoyl)phenyl]piperidine-1-carboxamide
8-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(2R,3R)-1'-(furan-3-carbonyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
5-{2-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid
1-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}piperidin-2-one
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
1-[2-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
9-(2-amino-6-methoxypyrimidin-4-yl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
(2-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}phenyl)methanol
(2E)-N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-2-yl)prop-2-enamide
N-{[5,8-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}cyclopentanamine
2-[1-(3-phenylpropyl)-4-(quinolin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-(2-methoxyethyl)-3-(2-methoxyphenyl)-3-{2-[(2S)-4-methyl-2-phenylpiperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2,7,8-trimethyl-4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]quinoline
2-cyclopropyl-4-hydroxy-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]pyrimidine-5-carboxamide
6-(benzyloxy)-4-(2-methoxy-2-phenylacetyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-[(2-propyl-1,3-thiazol-4-yl)methyl]thian-4-amine
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
(3S,4S)-1-(pyridin-4-ylmethyl)-4-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)pyrrolidin-3-ol
4-[1-(1-methylpiperidin-4-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]pyridine
1-(4-benzylpiperazin-1-yl)-3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]propan-1-one
2-phenoxy-N-{1-[7-(quinolin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
N-(adamantan-2-yl)-2-(1-benzyl-3-oxopiperazin-2-yl)acetamide
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-(2-{1-[2-(pyrrolidin-1-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
5-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}propan-1-one
(4aS,7aR)-1-[2-(dimethylamino)acetyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4-benzyl-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
N-(1-{1-[2-(4-methoxyphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
1-ethyl-N-[(1R)-1-(2-fluorophenyl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
3,5-difluoro-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
[(3R,4R)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-(2-phenoxyphenyl)benzamide
1-benzyl-4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
2-amino-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
4-(2-methoxyphenoxy)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
8-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-benzyl-1-ethyl-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-butanamido-N-(6-hydroxy-6-methylheptan-2-yl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
9-(cyclopropylmethyl)-1-methyl-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
[(2-{[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxy}phenyl)methyl]dimethylamine
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](2-methylpropyl)(pyridin-2-ylmethyl)amine