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2-(4-fluoro-3-methylbenzenesulfonamido)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
4-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}morpholine
2-(1H-1,3-benzodiazol-2-yl)-N-[3-(oxolan-3-yl)propyl]acetamide
2-methyl-7-(1,3-thiazol-4-ylmethyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-ethyl-4-pentanamido-N-(pyridin-4-ylmethyl)benzamide
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
5-ethyl-1'-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridine-3-carboxamide
(1S,5R)-3-(oxan-4-yl)-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-9H-purin-2-amine
2-(methylsulfanyl)-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-{2-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]ethyl}acetamide
9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-3-(quinolin-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-6-methylquinolin-4-ol
4-(5-{[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2,6-dimethyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]quinoline-4-carboxamide
(1s,4s)-4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)cyclohexan-1-ol
2-phenyl-1-(1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)ethan-1-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylbutanamide
2-{4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-1-(morpholin-4-yl)ethan-1-one
N-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
N-(adamantan-2-ylmethyl)-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(4-fluorophenoxymethyl)piperidine
N-(3-hydroxy-3-phenylpropyl)-N-methylquinoxaline-6-carboxamide
3,5-dichloro-4-methyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
3-[(4-fluorophenyl)methyl]-5-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
4-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]oxane-4-carboxylic acid
[1-(1-{[2-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-methylpyrimidine-5-carboxamide
2-methoxy-1-{4-[1-(9H-purin-6-yl)piperidin-4-yl]-1,4-diazepan-1-yl}ethan-1-one
[1-(4-fluorobenzoyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
3-(3-hydroxy-3-methylbutyl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide
(3S,4S)-1-(1H-1,3-benzodiazole-5-carbonyl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
(1S,5R)-3-(2-amino-6-methylpyrimidin-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[5-chloro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-(3-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-(4-methylphenyl)propan-1-one
2-(3-chlorophenoxy)-1-{4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}propan-1-one
5-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyridine-2-carbonitrile
(3S,4R)-1-(3,4-difluorobenzoyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
1-[(2-chlorophenyl)methyl]-N-methyl-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-5-(methoxymethyl)-1,3,4-oxadiazole
[(3R,4R)-1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(4aS,8aR)-1-butyl-6-(2-chlorobenzoyl)-decahydro-1,6-naphthyridin-2-one
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(4-methyl-1H-imidazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-oxoethyl]-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-one
2-[(5-methylpyrazin-2-yl)methyl]-8-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[(3S,4R)-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(2-fluorophenyl)pyridine-3-carbonitrile