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3-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
3-{4-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]phenyl}propanoic acid
2-[({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}amino)methyl]-5,8-dimethylquinolin-4-ol
N-[(4-phenyloxan-4-yl)methyl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
4-(furan-2-yl)-N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-benzyl-5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-ethyl-1,2-oxazole-3-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
9-(cyclohex-3-ene-1-carbonyl)-2-(furan-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2,4,5-trifluoro-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
ethyl 3-{2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamido}propanoate
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-(2-methylphenyl)-N'-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N'-(pyridin-2-ylmethyl)propanediamide
N-[2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-(thiophen-2-yl)butanamide
N-(1-{4-[(thiophen-2-ylmethyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
{[(3R,4S)-4-cyclopropyl-1-(2-phenoxyethyl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
(2S)-1-acetyl-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrrolidine-2-carboxamide
4-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-1-propylpyrrolidin-2-one
2-amino-8-[2-(pyrrolidin-3-yl)benzoyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(4-methyl-1H-pyrrole-2-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
(2R,4R)-N-{[3-(benzyloxy)phenyl]methyl}-4-hydroxypyrrolidine-2-carboxamide
1-(2,3-dimethoxyphenyl)-2-(3-ethynylbenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-[methyl(phenyl)amino]ethan-1-one
ethyl 4-{[1-benzyl-3-(dimethylcarbamoyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}piperidine-1-carboxylate
3-{[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole
4-ethenyl-N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
8-(1H-indol-5-ylmethyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-cycloheptyl-4-{4-[3-(2-oxopyrrolidin-1-yl)benzoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N,N-diethyl-1-[3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidine-3-carboxamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}[(1-methanesulfonylpiperidin-3-yl)methyl]amine
1-{5-[3-hydroxy-3-(hydroxymethyl)piperidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
{5-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-imidazol-2-yl]furan-2-yl}methanol
2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(thiophen-3-yl)phenoxy}-N-[(3,4,5-trimethoxyphenyl)methyl]acetamide
5-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-methyl-5-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(1S,5R)-3-(2-methyl-5-propylpyrimidin-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[3-cyclopentyl-5-(2-methyl-1H-1,3-benzodiazol-5-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
(2R,3R,6R)-3-(4-fluorophenyl)-5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(2-methoxyethyl)propanamide
2-[methyl({4-methyl-5-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-acetamido-1-ethyl-2-(3-methoxyphenyl)-1H-1,3-benzodiazole-7-carboxamide
4-chloro-6-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}-1H-pyrrolo[2,3-b]pyridine
1-(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}azetidin-3-yl)piperidine
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]azepan-3-amine
[2-(azepan-1-yl)ethyl]({[2-(methoxymethyl)pyrimidin-5-yl]methyl})(propan-2-yl)amine
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
methyl 5-{3-[benzyl(methyl)amino]piperidin-1-yl}-5-oxopentanoate
2-amino-6-cyclopropyl-4-(isoquinolin-5-yl)pyridine-3-carbonitrile