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8-[(2,3-dimethoxyphenyl)methyl]-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)(methyl)(pyridin-3-ylmethyl)amine
2-methyl-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)furan-3-carboxamide
5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
N-[(2R,3R)-2-ethoxy-1'-[(2-hydroxynaphthalen-1-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
(3R)-3,4,4-trimethyl-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]pyrrolidin-3-ol
1-(4,7-dimethylquinazolin-2-yl)-N-[(3,4,5-trimethoxyphenyl)methyl]piperidine-3-carboxamide
N-butyl-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-{[4-(propan-2-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({4-[2-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
4-{[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]methyl}-3,5-dimethyl-1-propyl-1H-pyrazole
5-(4-chloro-2-methoxyphenoxymethyl)-N-(2-methoxyethyl)-1,2-oxazole-3-carboxamide
5-{[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]isoquinoline
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}diethylamine
(4S)-4-amino-5-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-5-oxopentanoic acid
(1R,9aR)-1-({[(3,4-dimethoxyphenyl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
{5-[4-(2-amino-1,3-thiazol-4-yl)phenyl]-2-fluorophenyl}methanol
(5S,9aS,9bS)-5-(3,4-dimethylphenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-chloro-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2,5-dimethylbenzene-1-sulfonamide
1-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(5S,9aS,9bS)-5-(2,5-difluorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]methyl}-2,1,3-benzoxadiazole
N2,N2-dimethyl-N5-(1-propylpiperidin-4-yl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
5-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole
N-(2-{3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenoxy}propyl)pyridine-3-carboxamide
1-{4-[4-(azepane-1-carbonyl)phenoxy]piperidin-1-yl}-3-methoxypropan-1-one
(1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
(2S,4R)-4-{[(3-phenoxyphenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 1-{[3-cyclohexaneamido-2-(methoxycarbonyl)thieno[2,3-b]pyridin-6-yl]methyl}piperidine-3-carboxylate
2-benzyl-4-[3-(benzyloxy)azetidine-1-carbonyl]-1,3-thiazole
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]morpholine
4-{3-cyclopropyl-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}-2-methylpyridine
{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)[1-(pyridin-3-yl)ethyl]amine
2-({1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
2-(2-{[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
2-ethyl-7-(2-methoxybenzamido)-N-(2-methoxyethyl)-1-methyl-N-(propan-2-yl)-1H-1,3-benzodiazole-5-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-ethynylphenyl)methyl]piperidin-3-yl}propanamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-phenylpropanamide
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]propanamide
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
N-[3-(3-chlorophenyl)phenyl]-1-(3-methoxypropanoyl)piperidine-4-carboxamide
3-methyl-2-{4-phenyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-imidazol-5-yl}-1H-indole
2-{4-[3-(1-methoxyethyl)phenyl]phenoxy}-N-methylacetamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-3-methyl-2-phenylbutan-1-one
2-(3-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}piperidin-1-yl)pyrimidine
2-{2-[(dimethylamino)methyl]phenoxy}-6-methylpyridine-3-carboxamide