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5-{3-[4-(2-methylphenyl)piperazin-1-yl]-3-oxopropyl}-5-[(4-phenylphenyl)methyl]pyrrolidin-2-one
1-[(4-methylthiophen-2-yl)sulfonyl]-3-(3-methylthiophene-2-carbonyl)piperidine
2-benzyl-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-1,3-benzoxazole-5-carboxamide
2-hydroxy-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyridine-3-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-(1-acetylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-4-carboxamide
5-(4-chloro-1,5-dimethyl-1H-pyrazol-3-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-(4-chloro-1-methyl-1H-pyrrol-2-yl)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazole
N2-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(4-methylpyridin-2-yl)ethane-1,2-diamine
N-(cyclobutylmethyl)-2-[1-ethyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
8-[(3,5-difluorophenyl)methyl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R)-1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}pyrrolidine-2-carboxamide
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(oxan-2-yl)ethyl]amine
(1R,3S)-3-(2-aminoethoxy)-7-(propane-2-sulfonyl)-7-azaspiro[3.5]nonan-1-ol
({5-[1-(furan-3-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
ethyl 1-[(4-{[(5-methylfuran-2-yl)methyl]amino}quinazolin-2-yl)methyl]piperidine-3-carboxylate
(3R,4R)-4-(azepan-1-yl)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-ol
3-(1H-pyrazol-1-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
2-amino-4-ethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,3-thiazole-5-carboxamide
3-(1H-1,2,3,4-tetrazol-1-yl)-1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
(4aS,7aR)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(3,4-dichlorophenyl)-4-(2,3-dihydro-1-benzofuran-5-carbonyl)morpholine
9-methoxy-3-(2-methylpyridine-3-carbonyl)-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(2R,3R)-2-methoxy-1'-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
3-({5-[5-(oxan-2-yl)thiophen-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
N-cyclopropyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-cyclopentyl-N3-ethyl-N5-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-amino-8-(isoquinolin-5-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
4-(2-methoxyethyl)-1-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-(methoxymethyl)thiophene-2-carboxamide
1-(4-amino-5-cyanopyrimidin-2-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
1-(1-benzylpiperidin-4-yl)-N-methyl-N-(2-methylpropyl)piperidine-3-carboxamide
5-[(3-fluorophenyl)methyl]-5-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-3-(2-methylpropyl)imidazolidine-2,4-dione
6-tert-butyl-1-methyl-4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-1H-pyrazolo[3,4-d]pyrimidine
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(pentan-3-yl)-1,3-oxazole-4-carboxamide
N-(1-{7-[(2-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-3,5-dimethylbenzamide
ethyl 4-(2-{[2-(methoxycarbonyl)piperidin-1-yl]methyl}-8-methylquinazolin-4-yl)piperazine-1-carboxylate
6-methyl-2-{[4-(5-methyl-1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}pyridin-3-ol
N-[(4-fluorophenyl)methyl]-N-methyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carboxylic acid
N-[2-(2-fluorophenyl)-1-[1-(4-phenylbutanoyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
1-(furan-2-carbonyl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepane
6-(3,5-dimethoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
N-[(3R,4S)-4-cyclopropyl-1-(4-ethyl-5-methylpyrimidin-2-yl)pyrrolidin-3-yl]-2-hydroxyacetamide
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
N-{[1-(3-methylphenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]methyl}methanesulfonamide
N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-4-(pyrrolidin-1-yl)butanamide
N-ethyl-6-methoxy-2-oxo-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-[3-(2-methoxyphenyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine