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methyl 3-[(4-methoxyphenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-N-cyclohexyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(2-hydroxyphenyl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
3-[4-({[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-(thiophen-2-yl)butanamide
1-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-methoxyethan-1-one
N-cyclopropyl-3-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)propanamide
1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(2-ethoxyphenyl)piperazine
6-(piperidin-4-yl)-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)pyrimidin-4-amine
1-[(2,4-dimethoxy-3-methylphenyl)methyl]-3-(3-methoxybenzoyl)piperidine
4-(2-fluoro-5-methylphenoxy)-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxylic acid
4-[5-({3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}carbamoyl)pyridin-2-yl]benzoic acid
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
5-(2-methoxy-5-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazole
methyl (2S)-2-(3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-2-phenylacetate
2-[2-(azocan-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
{4-[2-(methylsulfanyl)benzoyl]-1,4-oxazepan-6-yl}methanol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-oxo-2-phenylacetyl)piperidine-2-carboxamide
5-[1-(1,1-dioxo-1λ6-thiane-4-carbonyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
2-[4-(1-benzothiophen-3-yl)-2-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy]-N-cyclopropylacetamide
methyl 4-(5-{[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
4-methyl-3-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
3-(2-oxopiperidin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
2-(1-ethyl-1H-1,2,4-triazol-5-yl)-1-methyl-1H-1,3-benzodiazole
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
[(2,3-dimethoxyphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-{4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}-3-phenoxypropan-1-one
8-[(3,4-dimethylphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(cyclopropylmethyl)({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})propylamine
(1R,3S,5S)-8-[4-(4-chlorophenoxy)piperidine-4-carbonyl]-8-azabicyclo[3.2.1]octan-3-ol
4-benzyl-3-ethyl-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,4-diazepan-5-one
3-{1-[5-(2-fluorophenoxymethyl)-1H-pyrazol-3-yl]-N-methylformamido}-N-methylbutanamide
methyl 3-(cyclohex-3-en-1-ylmethyl)-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2-methoxyethyl)-3-(propan-2-yl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
1-(4-benzylpiperazine-1-carbonyl)-6-{[4-(pyrrolidin-1-yl)phenyl]methyl}-6-azaspiro[2.5]octane
2-methyl-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-pyrrol-1-yl)propanamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butan-1-one
(1S,5R)-3-(3-methoxybenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{1-[2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]piperidin-3-yl}benzoic acid
1-{1'-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-[3-({[(4,6-dimethylpyrimidin-2-yl)methyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-methyl-5-phenylpiperidin-2-one
5-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-[(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)methyl]-1H-indazole-3-carboxamide