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2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[2-(hydroxymethyl)piperidin-1-yl]ethan-1-one
methyl 1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-3-phenylpyrrolidine-3-carboxylate
1-[2-(3-methoxyphenyl)ethyl]-2-(thiophen-3-yl)-1H-imidazole
5-{3-[4-(2-ethoxyphenyl)piperazin-1-yl]-3-oxopropyl}-5-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]piperidine-4-carboxamide
7-(2,8-dimethylquinoline-4-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-{[2-(difluoromethoxy)phenyl]methyl}-1-(4-methoxyphenyl)piperazin-2-one
5-ethyl-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1,2-oxazole-3-carboxamide
6-methyl-9-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-9H-purine
[(3R,4R)-1-(2-methylpyrimidin-4-yl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-5-hydroxy-4H-pyran-4-one
3-{5-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol
(4aS,8aR)-1-(carboxymethyl)-6-(1,3-thiazol-4-ylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]pyrrolidin-2-one
1-cyclopropyl-N-[(6-methylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
1-cyclohexyl-4-[2-(1H-indol-3-yl)acetyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
2-tert-butyl-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-4-hydroxypyrimidine-5-carboxamide
2-cyclopentanecarbonyl-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
7-(2-chloro-5-methylbenzoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrazol-3-yl)pyridine
2-(pentan-3-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(oxolane-2-carbonyl)-1,4-diazepane
1-benzyl-8-(2-methylbutyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{5-[3-(pyridin-4-yl)azetidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
2-{[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]methyl}-1,4-dihydroquinolin-4-one
N-(cyclopropylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(oxolan-2-ylmethyl)piperidin-4-amine
2-{4-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-3-(pyridin-4-yl)propanamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(5-methylpyrazin-2-yl)methyl]benzamide
3-methyl-1-(prop-2-en-1-yl)-4-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
3-{5-[(2-ethyl-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
ethyl 3-({2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxyphenyl}formamido)propanoate
N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
3-(2-{6-[(3-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
6-methyl-2-(2-{[3-(pyridin-3-ylmethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N,N-diethyl-1-[(1s,4s)-4-(5-phenoxyfuran-2-amido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3,4,7-trimethyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-indole-2-carboxamide
1-[2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetyl]-3-ethylpiperidine-3-carboxylic acid
N-[2-(2-chlorophenyl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
3,5-dimethoxy-2-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)benzoic acid
5-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)carbamoyl]amino}-2-methoxy-N,N-dimethylbenzamide
methyl 1-benzyl-3-cyclopropaneamido-5-{[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 1-{[4-(5-methoxy-5-oxopentanoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate