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methyl 1-ethoxy-2-oxo-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-(thiophen-3-ylmethyl)acetamide
5-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl)-3-methyl-1,2-oxazole
1-cyclopropyl-5-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}piperidin-2-one
(4aS,7aR)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[2-(aminomethyl)phenyl]benzonitrile
6-(cyclopropylmethoxy)-4-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl][(1-phenyl-1H-pyrazol-5-yl)methyl]amine
4-{2-[4-hydroxy-3-(prop-2-en-1-yl)phenyl]-1H-imidazol-1-yl}benzamide
(2E)-3-(4-chlorophenyl)-1-[1-(4-cyclohexylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]prop-2-en-1-one
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(methylsulfanyl)propyl]amine
2-(2-methyl-1,3-thiazol-4-yl)-N-{1-oxaspiro[4.4]nonan-3-yl}acetamide
N-{1-[1-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-(1-{2-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-2-oxoethyl}-1H-pyrazol-4-yl)furan-2-carboxamide
6-(benzyloxy)-1-cyclohexyl-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-1,4-diazepan-2-one
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(2-fluoropyridin-3-yl)urea
1-(pyridin-2-ylmethyl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
3-(1-{[2-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)-N-cyclopropylpropanamide
6-[1-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-3-yl]-2-methyl-3,4-dihydropyrimidin-4-one
N-(pyridin-3-ylmethyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
(3S,4S)-1-(2-amino-9H-purin-6-yl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
4-[2-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidin-2-amine
5-(1H-indol-1-ylmethyl)-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-3-carboxamide
4-benzyl-3-ethyl-1-(4-hydroxybenzoyl)-1,4-diazepan-5-one
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(6-methylpyridin-2-yl)methyl]amine
5-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-{[1-(2-methylphenyl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}methanesulfonamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-1-methyl-1H-pyrazole-5-carboxamide
N-ethyl-4-[3-(3-fluorophenyl)-1H-pyrazole-4-amido]piperidine-1-carboxamide
1-methyl-2-(morpholin-4-yl)-5-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1H-1,3-benzodiazole
ethyl 2-(1-{2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidin-2-yl)acetate
1,9-dimethyl-4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecane
N-methyl-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-(propan-2-yl)piperidin-4-amine
(1R,5S,6S)-6-({4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-4-(pyrrolidine-1-carbonyl)pyridin-2-amine
3-[(2,3-difluorophenyl)methyl]-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
6-methoxy-3-{[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[1-(pyridin-4-yl)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-(pyrrolidin-1-yl)pyrrolidine
3-(2-methoxyethyl)-1-[2-(morpholin-4-yl)-2-oxoethyl]piperidine-3-carboxylic acid
1-[7-(2-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl]-N,N-dimethylmethanesulfonamide
(3S,4S)-4-propyl-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidine-3-carboxylic acid
(2E)-3-(2,5-difluorophenyl)-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[3-(3-fluorophenyl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
2-ethyl-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)pyrimidine-5-carboxamide
3-(naphthalen-1-ylmethyl)-N-[2-(thiophen-2-yl)ethyl]-1,2-oxazole-5-carboxamide