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[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-indol-2-yl]methanol
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-(methoxymethyl)pyrimidin-4-amine
[2-(azepan-1-yl)ethyl](ethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
11-(5-ethoxyfuran-2-carbonyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-[(1-butyl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydro-1H-indazol-3-one
N-{[8-(1,3-benzothiazol-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propane-2-sulfonamide
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(1H-imidazol-2-ylmethyl)piperidine-3-carboxylic acid
3-{2-[4-(4-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}-1-cyclopropyl-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
4-phenyl-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-ol
2-chloro-4-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
4-{3-[4-(3-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
methyl 4-(5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-(prop-2-en-1-yl)-4-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrrolidin-2-one
5-(2-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-(3,3,5,5-tetramethylcyclohexyl)acetamide
6-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridin-3-ol
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
2-(2,3-dimethoxyphenyl)-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]acetic acid
4-{2-[4-(3-methoxybenzoyl)morpholin-3-yl]acetyl}piperazin-2-one
(1R,9S)-5-amino-12-methyl-3-[5-(1H-pyrazol-3-yl)furan-2-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]-2-{methyl[1-(1,3-thiazol-2-yl)ethyl]amino}acetamide
2-fluoro-N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-5-sulfamoylbenzamide
4-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-N,N-dimethylpiperazine-1-carboxamide
3-(2-aminoethyl)-4-(3,4-dimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-{[3-(furan-2-yl)phenyl]methyl}-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(2-methylpyridin-3-yl)oxy]-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
2-[(1S,5R)-6-(4-ethyl-5-methylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-[(3,4-dimethoxyphenyl)methyl]-2-(4-phenylpiperidin-1-yl)acetamide
(oxolan-2-ylmethyl)(pyridin-2-ylmethyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(3-methylbutyl)-8-(propan-2-yl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(8-methoxyquinolin-5-yl)methyl](methyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
2-[2-(pyridin-4-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
4-[2-({4-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-3-yl]-5-methylpyrimidin-2-yl}sulfanyl)ethyl]morpholine
N-[(2-chloro-5-fluorophenyl)methyl]-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
1-(azepan-1-yl)-3-[4-chloro-2-({[3-(dimethylamino)propyl]amino}methyl)phenoxy]propan-2-ol
2,6-dimethyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]quinoline-4-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-2-[4-(pyridin-4-yl)piperidin-1-yl]pyrimidine
N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-2-(1H-1,2,3-triazol-1-yl)acetamide
2-[({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)methyl]-3,5-dimethylpyridin-4-ol
6-chloro-N-cyclobutyl-2-(2-cyclopropylpyrimidin-5-yl)quinoline-4-carboxamide
6-ethyl-N-[(4-hydroxyphenyl)methyl]-2-oxo-N-(pyridin-3-ylmethyl)-1,2-dihydropyridine-4-carboxamide
ethyl 3-[2-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-5-oxopyrrolidin-1-yl]propanoate
2-(4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
2-(morpholin-3-yl)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethan-1-one
N-(2-{1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-2-yl}ethyl)acetamide
1-(2-aminoethyl)-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide