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1-{4-[methyl(prop-2-yn-1-yl)amino]piperidin-1-yl}ethan-1-one
5-methyl-5-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}imidazolidine-2,4-dione
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N,N-dimethyl-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
(5S,9aS,9bS)-5-[3-(2-methylphenyl)phenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{3-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
3-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-1-yl)-1,2-benzothiazole
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-(oxolan-3-yl)acetamide
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(3-methylphenyl)-3-{1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-4-yl}propanamide
3-hexyl-8-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamide
{1-[(2E)-3-phenylprop-2-en-1-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
2-[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazole
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
ethyl 4-{6-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-(3-methoxyphenyl)propanamide
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]butan-1-one
1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
5-acetyl-N-[2-(azepan-1-yl)-2-phenylethyl]thiophene-3-carboxamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]pyrrolidine-2-carboxamide
N-(1-benzylpiperidin-4-yl)-1-cycloheptyl-6-oxopiperidine-3-carboxamide
6-[5-(methoxymethyl)furan-2-carbonyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
N-(oxan-4-ylmethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-6-methyl-3-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(4-methoxy-3,5-dimethylphenyl)-1-(oxan-4-yl)urea
(2S,4S,5R)-1,2-dimethyl-4-[methyl(pyrazin-2-ylmethyl)carbamoyl]-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
N5-[1-(4-chlorophenyl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-[1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-phenoxypropan-1-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)cyclopropanecarboxamide
1-(4-methylpiperazin-1-yl)-3-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]propan-1-one
2-(1-ethylpiperidin-4-yl)-1-[4-(3-methylpyridin-4-yl)piperazin-1-yl]ethan-1-one
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-2-(4-methoxyphenyl)pyrimidine
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-1-methyl-3-phenyl-1H-pyrazole
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
5-[3-(methoxymethyl)piperidine-1-carbonyl]-2-(1-methyl-1H-pyrazol-4-yl)pyridine
N-cyclohexyl-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methylbenzamide
N-[4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}propanamide
3-[3-(2-chlorophenyl)propanoyl]-N-(furan-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(4-methylpiperazin-1-yl)-6-[2-(propan-2-yloxy)phenyl]pyrimidin-2-amine
N4-[2-(2,4-dimethoxyphenyl)ethyl]-5-ethylpyrimidine-2,4-diamine
3-[(3R,4S)-3-(4-cyanobenzamido)-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
4-methoxy-3,5-dimethyl-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]benzamide
N-(propan-2-yl)-1-[(1s,4s)-4-[3-(2-methoxyphenyl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(1-methylpiperidine-3-carbonyl)piperidine-4-carboxylic acid
N-(2-hydroxyethyl)-5-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide