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3-(3-methyl-1H-pyrazol-1-yl)-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
3-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(4-phenyloxan-4-yl)methyl]propanamide
2-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-ethyl-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyrimidine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(4-cyclohexylphenyl)-1-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)urea
4-benzyl-3-{1-[3-(dimethylamino)pyrazin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{3-[2-(benzylamino)-4-methyl-1,3-thiazol-5-yl]-1H-pyrazol-1-yl}ethan-1-ol
2-methyl-5-phenyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-{[4-(1-ethylpiperidin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(azepan-1-yl)-3-(3-{[(prop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(5-acetylthiophen-3-yl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
9-(2,5-difluorobenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(3-methoxypyrazin-2-yl)pyrrolidin-3-yl]methanol
ethyl 1-[(2-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]piperidine-4-carboxylate
1-[3-({[6-(propan-2-yl)pyridazin-3-yl]amino}methyl)pyridin-2-yl]piperidin-3-ol
1-(cyclopropylmethyl)-4-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
(2S,4R)-1-[(2-fluorophenyl)methyl]-N-[(4-methylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-{[(2S,5R)-5-(thiomorpholin-4-ylmethyl)oxolan-2-yl]methyl}benzonitrile
N-[2-methyl-1-(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]furan-3-carboxamide
1-{5-[(2,2-dimethylpyrrolidin-1-yl)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
1-[4-(4-methoxyphenyl)butan-2-yl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
2-methyl-3-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
(3S,9aR)-8-[(3-chlorophenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(3-ethynylbenzoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-2-methoxybenzamide
N-[2-(2-methoxyphenyl)ethyl]-1-{2-[4-(methylsulfanyl)phenyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
1-cycloheptyl-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazole
2-[(4-methoxyphenyl)methyl]-N-methyl-1,3-benzoxazole-6-carboxamide
3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
N-[(1-hydroxycyclohexyl)methyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]oxane-4-carboxamide
ethyl 1-(cyclopropylmethyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-[3-(pyridin-3-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-(2,5-difluorophenyl)piperidine-1-carboxamide
1-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(2,3-dimethylbenzoyl)-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
{1-cyclohexyl-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}(phenyl)methanol
1-[(3,4-dimethylphenyl)methyl]-4-[4-(1H-imidazol-1-yl)butanoyl]piperazin-2-one
N-benzyl-N-ethyl-3-(1-phenylethyl)-1,2-oxazole-5-carboxamide
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(2-methylphenoxy)piperidine
N-[2-(4-fluorophenyl)ethyl]-5-[1-(furan-3-ylmethyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
{3-[(2,4-difluorophenyl)methyl]-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-3-yl}methanol
3-({[(4-chlorophenyl)methyl]amino}methyl)-1-(cyclohexylmethyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
[(5-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-[4-(5-ethenylpyridin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one