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2-hydroxy-4-(methylsulfanyl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]butanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylfuran-2-yl)methyl]acetamide
N-[(2R,3R)-1'-(3-cyclohexylpropanoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)cyclopropanecarboxamide
5-methanesulfonyl-1'-[3-(methylsulfanyl)propyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-[2-(3-fluorophenyl)piperidine-1-carbonyl]-1,3-benzothiazole
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
3-fluoro-N-[1-(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
4-{1-[2-methyl-5-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-imidazol-2-yl}-2-(propan-2-yl)pyrimidine
(3aR,7aS)-2-[5-(methanesulfonylmethyl)pyridin-2-yl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-[(1S,2R)-2-[(5,6-dimethylpyrimidin-4-yl)amino]-1-hydroxypropyl]phenol
2-{9-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
methyl[2-(4-methyl-1H-pyrazol-1-yl)ethyl]{[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
7-(3-chlorophenyl)-4-(quinolin-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[1-(2,6-dimethoxypyridine-3-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(7-methyl-2-oxo-2H-chromen-4-yl)acetamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]acetamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]morpholine-2-carboxamide
3-fluoro-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
N-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
8-[3-(2-methylpropyl)-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-1-yl]quinoline
N,N-diethyl-1-{[1-(quinolin-6-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-cyano-5-fluoro-N-[1-(1H-pyrazol-1-yl)propan-2-yl]benzamide
1,3-dimethyl-N-{[3-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
N-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
4-[(2S)-1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]pyrrolidine-2-carbonyl]morpholine
N3-(3-hydroxy-2,2-dimethylpropyl)-1-[(2-methoxyphenyl)methyl]-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}pyrrolidin-3-yl]methanol
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1H-indole-5-carboxamide
4-(2-fluorophenoxy)-1-[4-(methylamino)pyrimidin-2-yl]piperidine-4-carboxylic acid
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl][(3-methoxyphenyl)methyl]methylamine
ethyl 2-[methyl({6-[methyl(2-phenylethyl)carbamoyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)amino]acetate
8-(4-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
1-(2-phenoxyethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
1-[(4-fluorophenyl)methyl]-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(2-cyclohexaneamido-5-methylphenyl)pyrazine-2-carboxamide
2-{4-[(2-aminopyrimidin-5-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-[(4-methoxyphenyl)methyl]-4-[2-(pyridin-2-ylsulfanyl)acetyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
6-[(2,4-dimethoxy-3-methylphenyl)methyl]-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
(benzylsulfamoyl)(pyridin-2-ylmethyl)amine
6-methyl-4-[4-(2,2,2-trifluoroethyl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
(1S,5R)-3-[(5-fluoro-2-methoxyphenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N,5,6-trimethyl-N-[2-(oxan-2-yl)ethyl]pyrimidin-4-amine