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3-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
3-cyclopropyl-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazole
5-methyl-3-(4-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenyl)-1,2,4-oxadiazole
methyl 3-cyclobutaneamido-5-{[(3,5-dimethoxyphenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(2-methoxyethyl)-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-methyl-N-[2-(2-propoxyphenyl)ethyl]piperidine-4-carboxamide
5-(3,4-difluorophenoxymethyl)-N-[(3-methoxyphenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
6-cyclopentyl-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(5-chloro-2-methoxyphenyl)methyl]-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methylacetamide
1-[(3S,4R)-1-[3-(2-methoxyphenyl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(dimethylamino)piperidin-3-yl]-N-(2-methoxyethyl)propanamide
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-(azepane-1-carbonyl)-1-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(2-methoxyphenyl)propan-1-one
1-{3-oxo-3-[2-(3-phenylpropyl)morpholin-4-yl]propyl}azepan-2-one
[(3-chloro-5-fluorophenyl)methyl][(1-ethyl-1H-pyrazol-4-yl)methyl]methylamine
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-3-(trifluoromethyl)benzene-1-sulfonamide
N-(2,5-dimethylphenyl)-3-[(2,4-dimethylpyrimidin-5-yl)formamido]propanamide
methyl (2R,4S)-4-hydroxy-1-[(1-methyl-1H-1,2,3-benzotriazol-5-yl)methyl]piperidine-2-carboxylate
4-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-indol-3-yl)acetamide
2-(2-{1-[(3-chloro-2-fluorophenyl)methyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-[5-(methoxymethyl)thiophene-2-carbonyl]-3-[(methylsulfanyl)methyl]piperidine
2-(benzyloxy)-N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]acetamide
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-4-(trifluoromethyl)pyridine
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
7-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-N-(1,2-oxazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[2-(methylamino)pyrimidine-5-carbonyl]-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
N-cyclopropyl-1-[1-(thiophene-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
methyl 3-[(4-methoxy-2,5-dimethylphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[4-(4-acetylpiperazine-1-carbonyl)piperidin-1-yl]-2-[2-(3-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[({1-[2-(thiomorpholin-4-yl)ethyl]-1H-pyrazol-4-yl}methyl)amino]-2,3-dihydro-1λ6-thiophene-1,1-dione
N-{1-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-1H-pyrazol-4-yl}-3-(2-methoxyphenyl)propanamide
7-(3-phenylpropyl)-2-(pyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
methyl 8-[(4-ethylphenyl)methyl]-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
(1S,5R)-6-(1,3-thiazol-4-ylmethyl)-3-(4,4,4-trifluorobutanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
3-{2-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-imidazole-2-carboxamide
(3S,5R)-1-benzyl-N3-butyl-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
3-cyclopropyl-1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylfuran-3-carboxamide
1-(2-methanesulfonylethyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-{1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-methoxy-3-methyl-1H-indole-2-carboxamide