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3-[(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)formamido]propanamide
(1H-imidazol-2-ylmethyl)[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
2-({2-[3-(propan-2-yloxy)phenyl]ethyl}amino)propan-1-ol
3-(1-phenylethyl)-N-[2-(thiophen-2-yl)ethyl]-1,2-oxazole-5-carboxamide
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-benzyl-4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-oxoacetamide
2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N,N-dimethylaniline
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
1-(4-{4-[3-(dimethylamino)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)-3-methoxypropan-1-one
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
1-(2-fluorophenyl)-4-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)piperazine
5-methoxy-2-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-1H-indole
9-methoxy-N-methyl-3-[(2-methylphenyl)methyl]-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-(pyridin-4-yl)pyrimidine
N-({8-[(2-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1H-indole-5-carboxamide
(2S,4R)-1-(furan-2-ylmethyl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
N-ethyl-6-[4-(2-methoxyethoxy)phenyl]pyridine-3-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-{[4-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(1H-pyrazol-1-yl)propanamide
4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidine
4-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-N,N-diethylbenzene-1-sulfonamide
7-methyl-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1H-indole
[2-(2-ethoxyphenoxy)ethyl](methyl)(quinoxalin-2-ylmethyl)amine
5-[(benzyloxy)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
N,2-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1-benzofuran-5-carboxamide
N-[(2-{4-[5-(methoxymethyl)thiophene-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-{4-[(2-fluorophenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-(1H-indol-3-yl)-6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
7-[(4-fluorophenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-benzyl-8-(1H-indol-3-ylmethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(piperidine-1-carbonyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
3-[(4-{1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)methyl]pyridine
N-(3,4-difluorophenyl)-3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
2-[(3,4-dimethoxyphenyl)methyl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
7-fluoro-3-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)-1-(2-phenylethyl)-1,2-dihydroquinolin-2-one
N,N-dimethyl-3-[4-(1H-pyrrole-2-carbonyl)piperazine-1-carbonyl]piperidine-1-carboxamide
2-fluoro-N-[3-(3-hydroxyazetidin-1-yl)-3-oxopropyl]benzamide
(2S,4S)-4-amino-1-[2-(benzyloxy)benzoyl]pyrrolidine-2-carboxylic acid
3-(2,2-dimethylpropanoyl)-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-fluoro-N-{[1-(1H-indol-3-ylmethyl)piperidin-3-yl]methyl}benzamide
2-[3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)benzenesulfonamido]-N-methylacetamide
5-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}isoquinoline
1-methyl-4-{[5-(1-phenoxypropyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
(2S,4S)-4-amino-1-{2-[(2,4-dimethylphenyl)carbamoyl]acetyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-[3-(4-{[(3,4-dimethoxyphenyl)methyl]amino}piperidin-1-yl)phenyl]-4-phenylbutanamide
(3R,5S)-N-[2-(dimethylamino)ethyl]-5-(morpholin-4-ylmethyl)-1-(2-phenylethyl)piperidine-3-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperazine