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3-{[4-(dimethylamino)oxan-4-yl]methyl}-1-[2-(2-fluorophenoxy)phenyl]urea
N-[2-(4-{[2-(4-chloro-2-methylphenoxy)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]cyclobutanecarboxamide
(3R,4S)-4-cyclopropyl-1-[4-(3-fluorophenyl)benzoyl]pyrrolidin-3-amine
(1R,9aR)-1-({methyl[(5-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
5-(morpholin-4-yl)-2-{[4-(trifluoromethoxy)phenyl]methyl}-2,3-dihydropyridazin-3-one
4-(2,3-dimethylbenzoyl)-1-(2-methylphenyl)piperazin-2-one
5-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
methyl 4-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-phenylethyl)piperidin-1-yl]methyl}benzoate
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}butan-1-one
4-{1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}quinoline
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methyl-1H-1,3-benzodiazole
N-cyclohexyl-4-oxo-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
2-(4-{[4-(5-methyl-1H-pyrazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
4-phenyl-N-[1-(1-{spiro[2.4]heptane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-4-methylpyrimidine-5-carboxamide
8-(3-chloro-5-fluorobenzoyl)-2-(3-methylbutyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
9-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)quinoline-2-carboxamide
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
N-[4-(4-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]-2-(4-methoxyphenyl)acetamide
methyl 8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
methyl 1-[(3S,5S)-5-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]carbamoyl}-1-{[5-(3-chlorophenyl)furan-2-yl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(dimethylamino)-1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-(2-methylphenyl)ethan-1-one
(3S,4S)-1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
[(3R,4R)-1-[(2-chloro-4-fluorophenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-{2-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1H-indol-2-one
1-benzyl-N-ethyl-5-[(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxamide
N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
(3aR,6aR)-2-cyclopentyl-5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[1-(methoxymethyl)cyclopropyl]methyl}acetamide
5-[benzyl(methyl)amino]-2-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
(3S,4R)-1-(1-aminocyclopropanecarbonyl)-4-(2H-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
1-[5-(3-methylthiophen-2-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
3-(3-chlorophenyl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}propanamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxypropyl)acetamide
9-(4-fluorobenzenesulfonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-4-(thiophen-2-yl)butan-1-one
3-(methoxymethyl)-5-({2-[2-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({2-[(2-methylquinolin-8-yl)oxy]ethyl})amine
3-hydroxy-3-{[(1H-indol-2-ylmethyl)amino]methyl}-1-(2-phenylethyl)piperidin-2-one
8-methoxy-N-methyl-N-[(2-methylpyridin-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1,9-dimethyl-4-[3-(1H-pyrazol-1-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecane
2-[(1R,3S,3aS,6aR)-3-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-5-ethyl-1-(hydroxymethyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
2-ethyl-8-(3-methanesulfonylbenzoyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(1R,3R)-3-aminocyclopentyl]-3-(1H-imidazol-2-yl)benzamide