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3-(2-{1-[2-(2-methoxyethyl)-1,3-benzoxazole-6-carbonyl]piperidin-2-yl}ethyl)phenol
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(ethylamino)pyrimidine-5-carboxamide
2-(3-{[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
2-{5-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
4-(1-methyl-1H-imidazol-2-yl)-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidine
N-[(4-methoxynaphthalen-1-yl)methyl]-N-(propan-2-yl)-1,4-dioxane-2-carboxamide
8-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
6-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]methanol
N-({7-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)cyclopropanecarboxamide
4-(1-benzothiophen-2-ylmethyl)-11-[(cyclopropylmethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(4-cyanophenyl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
N-methyl-2-(N-phenylmethanesulfonamido)-N-(quinolin-8-ylmethyl)propanamide
3-(2,5-difluorobenzoyl)-1-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidine
1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-phenylazepane
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl][3-(5-methylfuran-2-yl)butyl]amine
2-methoxy-1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
methyl 3-[({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}formamido)methyl]-5-propanamidobenzoate
N-{1-[1-(cyclopropylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
N-{[1-(2H-1,3-benzodioxol-5-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
2-(5-{2-oxo-1-oxaspiro[4.4]nonan-4-yl}-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl)acetamide
N-phenyl-3-{1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}propanamide
N-{2-[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
2-amino-1-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-methylpropan-1-one
2-{[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methyl}benzonitrile
[2-(3-methoxyphenyl)ethyl]({[6-(pyrrolidin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
4-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-4H-1,2,4-triazole
1-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-4-amine
3-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-5,6,7,8-tetrahydroquinoline
5-(naphthalen-1-ylmethyl)-5-{3-oxo-3-[4-(thiophen-3-ylmethyl)piperazin-1-yl]propyl}pyrrolidin-2-one
N-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-cyclopropyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}adamantane-1-carboxamide
3-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]-N-(1,3-thiazol-2-yl)propanamide
3-(2-hydroxyphenyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
N-(4-{1-[2-(2-hydroxyethyl)phenyl]-1H-imidazol-2-yl}phenyl)acetamide
1-[1-(3-phenylbutyl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-butyl-1-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]urea
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2-methylphenyl)methyl]piperidine
3-(1-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}azetidin-3-yl)pyridine
3-(2-methylpropyl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1,2-oxazole-5-carboxamide
2-[2-(3-chlorothiophene-2-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
2-(ethylsulfanyl)-5-{1-[(1-methylpyrrolidin-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
N-(2-methyl-1-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)pyridine-2-carboxamide
6-methyl-5-[5-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-2-(thiophene-2-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
2-{3-cyclopropyl-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl}pyridine
3-[(2,3-dimethoxyphenyl)methyl]-4-methoxy-N-methylbenzamide
2-(1-ethyl-1H-pyrazol-4-yl)-7,8-dimethyl-4-(2-methylpiperidine-1-carbonyl)quinoline
N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-2-oxo-2H-chromene-3-carboxamide
9-[(2-phenylpyrimidin-5-yl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one