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N-(1-{2-[4-(2-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)furan-2-carboxamide
N-(3-chloro-4-methoxyphenyl)-6-[2-(1H-indol-3-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
ethyl 5-{[(2,2-dimethyloxan-4-yl)amino]methyl}-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazole
(4aS,8aR)-6-(1H-imidazol-2-ylmethyl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
4'-(naphthalen-1-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
[1-({4-[3-(4-fluorophenyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-3-yl]methanol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,3-dimethyl-3-phenylbutanamide
2-[1-(2-hydroxybutyl)-5-(2-phenoxyphenyl)-1H-1,2,4-triazol-3-yl]acetamide
2-(dimethylamino)-N-(1-{7-[2-(4-methoxyphenoxy)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
2-{4-[(2-fluoro-4-methoxyphenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2R)-1-hydroxypropan-2-yl]-4-(quinolin-6-yloxy)piperidine-4-carboxamide
ethyl 1-(benzylcarbamoyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
1-({[(4-ethyl-1,3-thiazol-2-yl)methyl]carbamoyl}methyl)piperidine-4-carboxamide
6-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}naphthalen-2-ol
(2R)-2-amino-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)pentanamide
1-benzyl-6-(pyridin-2-ylmethoxy)-4-(1,3-thiazol-2-ylmethyl)-1,4-diazepan-2-one
1-(1-phenylcyclopentanecarbonyl)-1,4-diazepan-6-ol
9-methoxy-N-[(4-methoxyphenyl)methyl]-3-[2-(methylsulfanyl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-ethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide
1-(2-cyclohexylethyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-[methyl(phenyl)amino]ethan-1-one
[1-(2-amino-2-methylpropyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
N-[2-(benzyloxy)ethyl]-5,6-dimethylpyridine-3-carboxamide
6-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
6-methyl-2-{[4-(morpholine-4-carbonyl)piperidin-1-yl]methyl}quinolin-4-ol
4-(1-aminocyclopropanecarbonyl)-5-benzyl-1-(3-phenylphenyl)piperazin-2-one
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(2,3,4-trimethoxybenzoyl)-1,4-diazepan-2-one
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(2-phenylethyl)amine
8-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
4-[(2-phenyl-1H-imidazol-4-yl)methyl]-1λ6-thiomorpholine-1,1-dione
N-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
1-{4-[(5-hydroxypentyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
N2,N2,5,6-tetramethyl-N4-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)pyrimidine-2,4-diamine
N-[2-(2,4-difluorophenyl)-1-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]ethyl]-N-methylpropanamide
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
N-(2-{4-[(5-ethylpyridin-2-yl)methyl]morpholin-2-yl}ethyl)methanesulfonamide
1-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-3-ethylurea
5-benzyl-N-[2-(1H-imidazol-4-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-{[4-(hydroxymethyl)phenyl]methyl}-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
2-[(2-{methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]carbamoyl}phenyl)amino]acetic acid
1-[2-methoxy-4-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
4-(dimethylamino)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide