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N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-(3-chloropyridin-2-yl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
4-[1-(3-chloro-4-fluorobenzoyl)piperidin-4-yl]-5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidine
1-(5-acetyl-2-methoxyphenyl)-3-methyl-3-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]urea
1-cyclohexyl-N3-(2-methylpropyl)-4-oxo-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopropyl-N-{[7-fluoro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-5-methylthiophene-2-carboxamide
2-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}-6-methoxyphenol
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(1-methoxybutan-2-yl)benzamide
1-(2-phenylethyl)-8-(propan-2-yl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-(1H-pyrazol-1-yl)butan-1-one
3-{2-[2-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-(2,3-dihydro-1-benzofuran-7-yl)-2-methyl-5H,6H,7H-cyclopenta[d]pyrimidine
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(4-methylmorpholin-2-yl)ethyl]benzamide
N-cyclohexyl-2-ethyl-7-(2-methoxybenzamido)-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
9-(2,4-dimethylquinoline-7-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-{[(5-ethylpyrimidin-2-yl)amino]methyl}-1-(2-methoxyethyl)pyrrolidin-2-one
5-(3-cyanopyridin-2-yl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N,N-diethyl-6-[(oxolan-3-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
(3S,4R)-1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
1-(cyclohexylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
5-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]-1,3,4-oxadiazol-2-amine
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
1-(1-cyclohexylpiperidine-4-carbonyl)-4-(pyridin-3-ylmethyl)piperazine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(4,4,4-trifluorobutanoyl)pyrrolidin-3-yl]acetamide
2-{[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
3-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
N-({7-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
N-[2-(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
2-(4-acetylphenoxy)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)acetamide
3-ethyl-N-({7-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
2-({3-[cyclopentyl(prop-2-en-1-yl)carbamoyl]phenyl}amino)acetic acid
3-[3-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-oxopropyl]-3,4-dihydroquinazolin-4-one
(1S,5R)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-hydroxy-1-methyl-N-{3-[methyl(phenyl)amino]propyl}piperidine-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
N-[(5-chloro-1H-indol-2-yl)methyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-(4-methoxybenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[2-chloro-4-({4-[(ethylcarbamoyl)methyl]piperazin-1-yl}methyl)phenoxy]propanoic acid
3-(2-oxoimidazolidin-1-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
3-{5-[(5-chlorothiophen-2-yl)sulfonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-amino-3-ethyl-N-[3-(methylsulfanyl)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-hydroxy-N-methyl-2-(phenoxymethyl)pyrimidine-5-carboxamide
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
5-fluoro-N,3-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide