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N-[3-(furan-2-yl)phenyl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine-4-carboxamide
2-({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-1-ol
N-[2-(propylsulfanyl)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-(2-methylpropyl)-8-[4-(methylsulfanyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
2,6-dihydroxy-N-[3-(2-methoxyphenyl)propyl]benzamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2,3-dihydro-1H-inden-1-yl)-5-methoxybenzamide
N-[2-(6-methylpyridin-2-yl)ethyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-{1-[2-(2-acetyl-4,5-dimethoxyphenyl)acetyl]piperidin-3-yl}propanamide
methyl 4-(3-{1-[2-(dimethylamino)acetamido]-3-methylbutyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl)benzoate
4-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-(4-methoxyphenyl)-1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-amine
3-[3-({[(2,3-dimethoxyphenyl)methyl]carbamoyl}amino)phenyl]-N-methylpropanamide
4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-1,4-oxazepane
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
N-{3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}acetamide
2-amino-4-(4,5-dimethylfuran-2-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-(propan-2-yl)-1-[(1s,4s)-4-(2,2-dimethyloxane-4-amido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(4-methoxyphenyl)phenyl]-1-[(5-methylthiophen-2-yl)methyl]piperidine-3-carboxamide
1-[(2S,4R)-1-(9H-fluoren-2-ylmethyl)-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-(1-methylpiperidin-4-yl)piperazine
9-(1H-indol-6-yl)-6-methyl-9H-purine
ethyl 2-{1-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]piperidin-2-yl}acetate
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-1H-pyrazole-4-carboxamide
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-(3-propanoylpiperidin-1-yl)propan-1-one
N-(2-methoxyethyl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[(3-fluorophenyl)methyl]-N-(3-phenylpropyl)-1,2-oxazole-5-carboxamide
methyl 2-[(3-methylbutyl)sulfamoyl]-6-(quinolin-2-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-cycloheptyl-6-oxo-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-methyl-N-(pyridin-3-ylmethyl)benzamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
(2E)-3-(3,4-difluorophenyl)-N-{[8-(4-fluorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}prop-2-enamide
1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
methyl 5-[(2S)-2-amino-3-(1,3-thiazol-4-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-(azocan-1-yl)-3-(2-methoxy-4-{[(2-phenylethyl)amino]methyl}phenoxy)propan-2-ol
(3R,4S)-4-{4-[(8-chloroquinolin-2-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
1-[1-(2-fluorophenyl)piperidin-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)urea
5-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
methyl 3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[3-(1H-indol-3-ylmethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]benzoic acid
N,N-diethyl-1-{[4-(phenylamino)quinazolin-2-yl]methyl}piperidine-4-carboxamide
(1R,2S,6R,7S)-4-(1H-indole-6-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
1-[(5-ethylpyridin-2-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
(3aS,6aS)-2-cyclopentanecarbonyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-fluoropiperidine
N-[(3R,4S)-1-acetyl-4-phenylpyrrolidin-3-yl]cyclopropanesulfonamide
N'1-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclopropane-1,1-dicarboxamide
N-cyclopentyl-2-ethyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}butanamide