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3-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
(3R,4R)-4-methyl-3-(propan-2-yl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-3-ol
1-[3-(dimethylamino)phenyl]-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
3-{[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)pyridine
1-{5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-4-(3-methylpyridin-4-yl)piperazine
1-[(2,5-dimethoxyphenyl)methyl]-3-(5-fluoro-2-methoxybenzoyl)piperidine
1,2-dimethyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1H-imidazole-4-sulfonamide
1-{4-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidin-1-yl}ethan-1-one
4-(2-hydroxy-4-methylpentanoyl)-1-(3-methoxyphenyl)piperazin-2-one
3-phenyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1,2-oxazole-5-carboxamide
1-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)-3-(4-methylphenyl)propan-1-one
2,8-dimethyl-N-[1-(1,3-thiazol-5-yl)propan-2-yl]quinoline-4-carboxamide
5-(2-methoxyacetamido)-1-methyl-N-(2-methylpropyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
2-methoxy-4-({[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
6-[6-hydroxy-4-(5-methyl-2H-1,2,3-triazole-4-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(6-methylpyridazin-3-yl)piperazin-2-yl}ethan-1-ol
1-butyl-4-(2-oxo-1-phenyl-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)piperazine-2,3-dione
1-(1,2-oxazinan-2-yl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-(1H-imidazol-2-yl)-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}piperidine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(pyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
5-[({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-ethyl-5-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-phenyl-1,2-oxazole-5-carboxamide
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylcyclohexane-1-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[3-(1H-indol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2,5-dimethyl-1-phenyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrrole-3-carboxamide
1-cyclobutanecarbonyl-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
3-{[4-(diethylamino)phenyl]methyl}-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{[4-(4-methoxyphenyl)piperazin-1-yl]methyl}-4-(pyridin-2-yl)phenol
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
5-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-2-(thiophen-2-yl)pyrimidine
3-[2-(4-acetyl-4-phenylpiperidin-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
methyl({[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl})[(4-phenyl-1,3-thiazol-2-yl)methyl]amine
1-[1-(4-chlorobenzoyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(1,3-thiazol-2-yl)acetamide
3-[1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-ethyl-1,2-oxazole-3-carboxamide
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-4-(benzyloxy)butan-1-one
1-[1-(dimethylamino)propan-2-yl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
5-{1-[2-(4-chloro-2-methylphenoxy)acetyl]piperidin-4-yl}-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(thiophen-2-ylmethyl)piperazine
1-{[2-(2-fluoro-5-methoxyphenyl)phenyl]methyl}piperazine
2-methyl-N-[phenyl(pyridin-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
methyl 5-[3-(pyridin-3-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-{3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(2-methoxyphenyl)propan-1-one