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2-(1-benzyl-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
8-fluoro-N-[2-(pyridin-2-ylsulfanyl)ethyl]quinoline-2-carboxamide
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
{3-[2-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]propyl}dimethylamine
4-{[4-(pyrrolidine-1-sulfonyl)-1,4-diazepan-1-yl]methyl}-2,1,3-benzoxadiazole
(3R,4R)-4-ethyl-1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperidine-3,4-diol
N-[4-(methylsulfanyl)phenyl]-6-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(oxan-2-yl)ethyl]amine
(2S,4S)-4-amino-N,N-diethyl-1-(4-methyl-1H-imidazole-5-carbonyl)pyrrolidine-2-carboxamide
ethyl 1-(2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetyl)piperidine-3-carboxylate
N-[2-(ethylsulfanyl)ethyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-cyclohexyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(propan-2-yl)acetamide
N-({3-[(4-fluorophenyl)methyl]phenyl}methyl)acetamide
2-(dimethylamino)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
8-[2-(cyclopent-2-en-1-yl)acetyl]-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-oxo-1-phenyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-2,5-dihydro-1H-pyrazole-3-carboxamide
(3aR,5R,6S,7aS)-2-{[3-(3-methoxyphenyl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
3-{[(2,2-difluoroethyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
1-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-methylbutan-1-ol
1-{1-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
3-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-2-yl}pyridine
(2S,4R)-4-amino-1-[2-(1H-imidazol-2-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(8R,9aS)-8-hydroxy-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
2-(dimethylamino)-N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-4-methylpyrimidine-5-carboxamide
2-(pyridin-4-yl)-4-(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)pyridine
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N,N-dimethylacetamide
1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)piperidin-3-ol
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-methoxy-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
4-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-6-methoxy-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
(4S)-4-amino-5-{2-cyclobutyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-5-oxopentanoic acid
methyl 3-(furan-3-amido)-5-({[4-(4-methylpiperazin-1-yl)phenyl]formamido}methyl)benzoate
2-[(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]ethan-1-ol
methyl 1-[(3S,5S)-1-[(4-fluorophenyl)methyl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 2-{1-[2-(4-methoxyphenyl)ethyl]-2,4-dioxo-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
methyl 4-({[6-oxo-1-(3-phenylpropyl)piperidin-3-yl]formamido}methyl)benzoate
1-[2-(benzyloxy)ethyl]-3-(1-ethyl-1H-imidazol-2-yl)piperidine
(4aS,8aS)-2-cyclopentanecarbonyl-7-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
(3R,5S)-5-[1-(2,3-dihydro-1H-inden-4-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-3-ol
N-[2-(1H-indol-1-yl)ethyl]-3-(2-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
ethyl 4-[3-(trifluoromethyl)-1H-pyrazole-5-amido]piperidine-1-carboxylate
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-ethoxyacetyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[5-(methoxymethyl)thiophene-2-carbonyl]pyrrolidin-3-yl]methanol
1-cyclobutanecarbonyl-3-[2-(3-methoxyphenyl)ethyl]piperidine
1-(2-fluorophenyl)-3-(propan-2-yl)-5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole