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4-{6-oxo-2,7-diazaspiro[4.5]decan-2-yl}butanoic acid
3-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
7-[(2-fluorophenyl)methyl]-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-3-(2-methylpropyl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,2-oxazole-5-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(4-fluorophenoxy)piperidin-1-yl]ethan-1-one
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(propan-2-yl)piperidin-4-amine
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]phenyl}-2-methylbutan-2-ol
3-(3-{[ethyl(oxolan-2-ylmethyl)amino]methyl}-1H-indol-1-yl)propanamide
N-benzyl-N-(2-hydroxyethyl)-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]acetamide
(2S,4S)-4-{[(2,6-difluorophenyl)methyl]amino}-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-2-carboxamide
1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}ethan-1-one
6-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
3-[4-(2,3-dichlorophenyl)piperazine-1-carbonyl]-2,8-diazaspiro[4.5]decane
N-(2-{4-phenyl-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}ethyl)acetamide
9-[(2,3-dimethoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-(2,3-dihydro-1H-inden-5-yl)-2-(3-fluorophenyl)-3-oxopiperazine-1-carboxamide
7-(furan-2-ylmethyl)-N4-[(1-methyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(4-methoxyphenyl)-3-phenylpropanamide
1-benzyl-N-[(2-chlorophenyl)methyl]-5-methanesulfonamido-2-methyl-1H-1,3-benzodiazole-7-carboxamide
6-[(2-fluorophenyl)methoxy]-4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-1-(2-methylpropyl)-1,4-diazepan-2-one
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[3-(pyridin-2-yl)propanoyl]-1,4-diazepan-2-one
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-[(2,3-difluoro-4-methylphenyl)methyl]-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{4-[(3,5-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-methylbutan-1-ol
[(3S,5R)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-N-methylpyridine-3-carboxamide
3-butanamido-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
1-[1-(2,8-dimethylquinoline-4-carbonyl)piperidin-4-yl]pyrrolidin-2-one
4-[1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenol
[1-(2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)piperidin-2-yl]methanol
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-cyclopropyl-2,3-dimethoxy-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}benzamide
2-(2-aminoethyl)-N-[(2,6-dimethoxyphenyl)methyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
4-acetamido-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]oxolane-2-carboxamide
4-({4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)morpholine
ethyl 1-(oxolane-2-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-2H-chromen-2-one
1-benzyl-4-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3-(thiophen-3-yl)propan-1-one
2-(2-chlorophenyl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(azocan-1-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
5-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}-N-(propan-2-yl)pyrimidin-2-amine