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N-[2-(1H-pyrazol-1-yl)ethyl]-7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(oxolan-2-ylmethoxy)acetamide
2-chloro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-5-(trifluoromethyl)benzamide
3-(1H-1,3-benzodiazol-2-yl)-N-[(1S,2R)-2-{[1-(propan-2-yl)piperidin-4-yl]amino}cyclobutyl]propanamide
N-[1-(3-methylphenyl)piperidin-4-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-benzyl-4-(1-methyl-1,2,3,4-tetrahydroquinoline-6-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-[1,3-dioxo-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)piperidine-4-carboxamide
2-[(3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}phenyl)amino]acetic acid
7-[ethoxy(phenyl)methyl]-4-[(3-methylquinoxalin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2-methylpropyl)-2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
N-[(3R,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
(3S,4S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-(naphthalen-2-yl)piperidin-3-ol
1-{2-[methyl({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl})amino]ethyl}piperidin-2-one
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2,2,2-trifluoroethyl)acetamide
1-{4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]piperidin-1-yl}ethan-1-one
2-(5-acetylthiophen-3-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-(2-cyclobutyl-1-methyl-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-1,3-benzodiazol-7-yl)oxolane-2-carboxamide
1,5-dimethyl-4-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(2S,4S)-4-cyclopentaneamido-N,N-diethyl-1-(furan-3-carbonyl)pyrrolidine-2-carboxamide
1-(cyclohexylmethyl)-N-methyl-5-{[2-(propan-2-yloxy)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(cyclohex-3-en-1-ylmethyl)(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-[2-(3-fluorophenyl)ethyl]-2-(4-{4-[(6-hydroxy-6-methylheptan-2-yl)amino]piperidin-1-yl}phenyl)acetamide
5-(4-fluorophenyl)-N-(3-methoxypropyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
4,6-dimethyl-1-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amine
4-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)-2-(propan-2-yl)pyrimidine
4-[3-(2-chlorophenyl)propanoyl]-1-(4-methoxyphenyl)piperazin-2-one
1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[1-(4-fluorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
7-methoxy-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,6S)-9-methyl-3-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
5-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
methyl 3-(2H-1,3-benzodioxol-5-ylmethyl)-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
9-(2-hydroxybutanoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-fluoro-3-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,4-dihydroquinolin-4-one
1-(cyclohexylmethyl)-6,7-dimethoxy-3-({[(4-methylphenyl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
4-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-2-amine
3,6-dimethyl-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-[3-(methylsulfanyl)propyl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-[(2-fluorophenyl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
5-(2-methoxyethyl)-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(cyclopropylmethyl)-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)-N-propylacetamide
1-benzoyl-N-[1-(thiophen-2-yl)propyl]piperidin-4-amine
2-(5-chloro-2-ethoxyphenyl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
3-(pentan-2-yl)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-chlorophenyl)-3-{1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}propanamide
3-methoxy-1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}propan-1-one
methyl (2S)-3-(4-hydroxyphenyl)-2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)propanoate