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2-[2-(tert-butylsulfamoyl)phenyl]-N-(propan-2-yl)pyridine-4-carboxamide
3-(oxolan-3-yl)-5-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-1,2,4-oxadiazole
4-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(1H-indol-1-yl)propyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[(1R)-1-(4-methoxyphenyl)ethyl]-2-(3-methylbenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-{2-[({thieno[3,2-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
2-(2-methyl-1,3-thiazol-4-yl)-N-{[8-(pyridin-3-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
N-{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)-2-methylpropanamide
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-1-(1-benzothiophen-2-ylmethyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
7-[(2-fluorophenyl)methyl]-2-[3-(1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-(4-chloro-2,5-dimethylbenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
3-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]urea
4-{2-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}-1λ6-thiomorpholine-1,1-dione
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]amine
(2R,6S)-4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
2-(dimethylamino)-N-{3-methyl-1-[7-(4-phenylbutanoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
2,4-dimethyl-N-{3-[methyl(phenyl)amino]propyl}-1,3-oxazole-5-carboxamide
N-[2-methyl-1-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]pyridine-2-carboxamide
6-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-6-(piperidin-3-yl)pyrimidin-4-amine
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(naphthalen-1-ylmethyl)amine
N-methyl-2-(methylsulfanyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-(2-methyl-1,3-thiazole-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
[2-ethoxy-5-({3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}methyl)phenyl]methanol
1-methyl-3-(naphthalen-2-ylmethyl)-8-(quinolin-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 9-(benzyloxy)-3-[(3-chlorophenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-ethyl-4-hydroxy-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-5-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
4-{6-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
2-(methylsulfanyl)-5-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyrimidine
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(2,3,4-trimethoxyphenyl)methyl]amine
N-(2-methoxyethyl)-1-[1-(quinolin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
4-[(2,3-difluorophenyl)methyl]-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-amine
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-(pyridin-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
(2R,3R,6R)-5-(2-methylpyrimidine-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-methyl-2-phenyl-6-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]pyrimidine
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-[(3S,4R)-1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(3-benzyl-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol
1-cyclohexyl-4-[3-(1H-indol-3-yl)propanoyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
7-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-5-propylpyrazolo[1,5-a]pyrimidine
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide