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N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-ethyl-N,5-dimethyl-1H-pyrazole-4-carboxamide
(1R,3S)-3-methoxy-7-[6-(morpholin-4-yl)pyrimidin-4-yl]-7-azaspiro[3.5]nonan-1-ol
3-(4-methoxyphenyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-phenylpropanamide
N-(1,4-dioxan-2-ylmethyl)-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
1'-(5-methyl-1,2-oxazole-3-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-amino-4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-7-methyl-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-3-methylpiperidine
N-ethyl-3-{[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]sulfamoyl}-N-methylbenzamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
4-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}-1λ6-thiomorpholine-1,1-dione
4-(2,6-dimethoxypyridine-3-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-[2-(2,4-difluorophenyl)-1-[1-(4-methoxybenzoyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)-4-(trifluoromethyl)benzamide
N,N-diethyl-1-[(1s,4s)-4-[(2E)-3-(thiophen-2-yl)prop-2-enamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(oxolan-3-yl)propyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-amine
4-[2-(2-methoxyphenoxy)acetyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-{3-[(2-chlorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}azepane
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(oxan-4-yl)pyrrolidine-2-carboxamide
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-4-(pyridin-2-yl)pyrimidin-2-amine
1-ethyl-3-methyl-N-[2-(pyridin-3-ylformamido)ethyl]piperidine-3-carboxamide
3-(2-methylphenyl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-6-fluoro-1H-1,3-benzodiazole-2-carboxamide
3-[({1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}oxy)methyl]pyridine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
5-(oxolan-3-ylmethyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-{2-[1-(quinoline-8-carbonyl)piperidin-2-yl]ethyl}phenol
N-(oxolan-2-ylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-(2-oxo-2-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}ethyl)pyrrolidin-2-one
1-(4-chloro-2,6-dimethylphenyl)-3-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}urea
7-[(3-methoxyphenyl)methyl]-2-(2-methoxypyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)propanamide
ethyl 1-benzyl-5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2E)-1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-3-(4-methoxyphenyl)prop-2-en-1-one
5-[1-(but-2-ynoyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
(3aS,6aS)-2-methyl-5-[(1-methyl-1H-indol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-diphenylacetamide
dimethyl(3-{2-[1-(2-methyl-1,3-benzoxazole-6-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
5-[4-(cyclopentylmethyl)piperazine-1-carbonyl]-1-(pyridin-2-ylmethyl)piperidin-2-one
2-phenyl-1-[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]ethan-1-one
[(3aS,6aS)-2-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
6-[4-(furan-2-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]pyridine-2-carboxamide
N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-4-methoxy-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-{2-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-4-carboxylic acid
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidin-3-yl]methanol
2-(2-phenylethyl)-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
2-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}benzoic acid