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5-(2-methoxy-2-phenylacetyl)-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(2-{4-[(dimethylamino)methyl]thiophen-2-yl}-1H-imidazol-1-yl)methyl]benzoic acid
N-[5-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)thiophen-2-yl]acetamide
5-(2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-(3-fluorophenyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-({7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methylbutanamide
2-(dimethylamino)-N-(1-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-N-methylacetamide
N-[(2-chlorophenyl)methyl]-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-(2-methylpropyl)benzamide
4-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
4-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,2-dimethylpiperazine
methyl 4-[(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]benzoate
ethyl(propan-2-yl)({1-[1-(propane-1-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
4-(1-ethyl-5-oxopyrrolidine-3-carbonyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-1,2,3-triazole-5-carboxamide
1-[4-(3-methoxyphenyl)piperazin-1-yl]-3-[(3S,4R)-1-(2-methylpropyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-one
(4aS,7aR)-1-(2-aminoacetyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-methoxy-N,N-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-ethyl-9-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
9-methoxy-3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2R,4R)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-4-hydroxy-N-methylpyrrolidine-2-carboxamide
N-[1-(oxan-4-yl)piperidin-4-yl]-2-(1H-pyrazol-1-yl)butanamide
5-{3-[4-(2-fluorophenyl)piperazin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
7-(1,3-benzothiazol-2-yl)-4-[(2-ethoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1,3-dimethyl-1H-pyrazol-4-yl)-4-[3-(morpholin-4-yl)-3-oxopropyl]piperidine-1-carboxamide
(butan-2-yl)[(6-methoxypyridin-3-yl)methyl](pyridin-4-ylmethyl)amine
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(2R,3R)-3-{[(2-chlorophenyl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
ethyl 4-[6-(1-methyl-1H-indole-2-carbonyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
1-(4-methoxypyrimidin-2-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-{[7-(3,4-dimethylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-fluorobenzamide
1-(oxane-4-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
7-methoxy-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydronaphthalen-2-amine
1-methyl-5-(2-phenylphenyl)-1H-imidazole
5-cyclopropyl-N-[3-(dimethylamino)propyl]-N-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-({4-[(4-acetamidophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-N,N-diethylpiperidine-3-carboxamide
5-[1-(1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-2-yl]-N,N-dimethylthiophene-2-carboxamide
2-methyl-N-(1,2-oxazol-3-ylmethyl)imidazo[1,2-a]pyrimidine-3-carboxamide
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(2-methylphenyl)piperidine-1-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
(2E)-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethylpent-2-enamide
N-[(2R,3R)-2-hydroxy-1'-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
2-(2-aminopyrimidin-5-yl)-N-ethyl-8-methyl-N-[2-(pyridin-2-yl)ethyl]quinoline-4-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(3-methylphenoxy)ethan-1-one
(2S)-N-{2-[(2,6-dimethylphenyl)carbamoyl]phenyl}oxolane-2-carboxamide
4-benzyl-2-{2-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
3,5-dimethyl-N-{3-methyl-1-[7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
2-(2-methoxyethyl)-9-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}phenyl)acetamide
methyl 3-{[1-(cyclopropylmethyl)-5-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide