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3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
2-(3-chlorobenzoyl)-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
N-({7-[(3,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-oxopyrrolidine-2-carboxamide
3-{[1-cyclohexyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})(quinoxalin-2-ylmethyl)amine
{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-2-yl}methanol
2-[3-(methylsulfanyl)phenyl]-3-(pyrrolidine-1-carbonyl)pyridine
(3R,4R)-1-[4-(5-methylfuran-2-yl)benzoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(pyridin-4-yl)-1,4-diazepan-6-ol
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4-methylpiperazine
1-{1-methyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-(1,3-thiazol-4-yl)ethan-1-one
methyl (2S)-1-{1-[4-({[2-(2-methoxyphenyl)ethyl]carbamoyl}methyl)phenyl]piperidin-4-yl}pyrrolidine-2-carboxylate
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
2-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-1,2-dihydroisoquinolin-1-one
2-{3-cyclopentyl-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-1-yl}benzoic acid
1-{1'-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
(3R,4R)-1-(5-ethyl-2-methylpyrimidin-4-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
methyl 3-acetamido-5-{[(3-fluorophenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}piperidine-4-carbonitrile
2,3,6-trimethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}quinoline-4-carboxamide
2-[(3-methoxyphenyl)methyl]-8-[2-(propan-2-ylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(4-chlorophenoxy)-N-(furan-3-ylmethyl)-N-methylpiperidine-4-carboxamide
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
N,N-dimethyl-4-[3-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidine-1-sulfonamide
(4aS,7aR)-N-cyclopentyl-4-[2-(dimethylamino)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-fluorobenzamide
3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-(4-fluorophenyl)urea
methyl 3-(2-methylbenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(1-{[1-(furan-2-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
6-[(2,4-difluorophenyl)methyl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
ethyl 4-{[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]amino}piperidine-1-carboxylate
N-[4-(4-{[(4-fluorophenyl)methyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
N-[1-(thiophen-2-yl)butyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 5-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}pyridine
1'-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-(2-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
N-[3-(cyclohexylsulfanyl)propyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-benzyl-N-methyl-3-[1-(oxane-2-carbonyl)piperidin-4-yl]propanamide
(4aS,7aR)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3S,5R)-1-(5-methoxyfuran-2-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
3-[5-(1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2-[(1-acetylpiperidin-4-yl)oxy]-N-[1-(4-chlorophenyl)ethyl]-5-methoxybenzamide
2-{3-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}-1,2-oxazinane
6-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carboxylic acid
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
N-({5-methyl-2-[3-(2-methylfuran-3-amido)phenyl]-1,3-oxazol-4-yl}methyl)-2-(propan-2-yl)oxane-4-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)-2-(pyridin-2-ylsulfanyl)acetamide