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2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
4-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-[5-(4-acetylpiperazine-1-carbonyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-3-cyclohexylpropanamide
2-(3-hydroxypropyl)-8-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-N-(piperidin-4-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{3-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}piperidine-4-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-(3-methoxypropyl)piperidine
2-methyl-N-(4-{[(2R)-pyrrolidin-2-ylmethyl]carbamoyl}phenyl)furan-3-carboxamide
(isoquinolin-5-ylmethyl)(methyl)[(5-methylfuran-2-yl)methyl]amine
3-[1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
3-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
(3aS,6aS)-2-(dimethylcarbamoyl)-5-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]phenyl}-1,3-diazinane-2,4-dione
1-[2-(ethylsulfanyl)phenyl]-3-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}urea
N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-2-(2-methyl-5-oxopyrrolidin-1-yl)acetamide
3-hydroxy-1-(2-phenylethyl)-3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}piperidin-2-one
methyl (2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-[(pyrimidin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
3-methoxy-1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydropyridin-2-one
N-[7-(3-hydroxypiperidine-1-carbonyl)-1-(2-methoxyethyl)-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,1,7-trimethyl-1H-indole-2-carboxamide
(4aS,8aR)-6-[2-(2,5-dimethylphenyl)acetyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
[(3S,5R)-1-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
methyl (2S)-1-[3-(3-chlorothiophene-2-carbonyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
N-{3-oxo-3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propyl}acetamide
4-(5-ethyl-2-methylpyrimidin-4-yl)-1-[(4-methylphenyl)methyl]piperazin-2-one
2-(3-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}phenoxy)ethan-1-ol
2-{3-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}-1,2,3,4-tetrahydroisoquinoline
6-[(5-methylthiophen-2-yl)methyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
ethyl 1-(3-acetyl-1H-pyrazole-5-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
ethyl 4-{4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}piperidine-1-carboxylate
(1-{1-[(3-chlorophenyl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
3-ethyl-5-methyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,2-oxazole-4-carboxamide
3-[(3R,4S)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-1,8-naphthyridine
{1-methyl-5-[2-(phenylamino)pyrimidine-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
7-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methylpropyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
6-chloro-N-[cyclopropyl(3-methylpyridin-2-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
8-(furan-3-ylmethyl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-cyclopentyl-N-(2-methoxyethyl)acetamide
5-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)pyrrolidin-2-yl]-N-ethylthiophene-2-carboxamide
7-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]-2-oxa-7-azaspiro[4.5]decane
3-(2-methoxyethyl)-8-methyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-(2-fluorophenyl)-5-[1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-{[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]amino}-6-methylpyridine-3-carboxamide
3-[4-(pyridin-3-yl)piperazine-1-carbonyl]-6-(trifluoromethyl)pyridin-2-ol