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4-{[2-(3-methoxy-6-methylpyridin-2-yl)phenyl]methyl}morpholine
4-ethyl-3-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4R)-1-[1-(2-fluorophenyl)piperidin-4-yl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,9-diazaspiro[5.5]undecane
1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
5-({3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{4-[(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazol-5-yl)methoxy]phenyl}-1H-1,2,4-triazole
N-[(2-methoxyphenyl)methyl]-2-(methylamino)-N-(propan-2-yl)acetamide
3-chloro-N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
2-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]pyridine-4-carboxamide
N-[(2S,4R,6S)-2-benzyl-6-(quinoxalin-2-yl)oxan-4-yl]acetamide
N-{[7-(2,3-dimethyl-1H-indole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
6-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(5-methylthiophen-2-yl)methyl]amine
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
methyl({[3-(1H-pyrazol-4-yl)phenyl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
6-(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-3-yl)-2-methyl-3,4-dihydropyrimidin-4-one
4-[(4-fluorophenyl)methyl]-1-(3-methyl-1,2-oxazole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(2E)-3-(2-chlorophenyl)-N-cyclopentyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)prop-2-enamide
2-(1-benzofuran-2-yl)-2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]quinoline
3-cyano-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
4-(2-fluoro-5-methylphenoxy)-1-(propylcarbamoyl)piperidine-4-carboxylic acid
2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
N-(3-fluorophenyl)-6-{[4-(furan-2-yl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}dimethylamine
N-cyclooctyl-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-(2-cyclopentylacetamido)-1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
3-benzyl-5-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1,2,4-oxadiazole
2-oxo-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1,2-dihydroquinoline-4-carboxamide
methyl 7-oxo-3-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-methyl-2-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
3-(3,4-dimethylphenyl)-1-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)propan-1-one
2-{1-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
1-cyclopropyl-5-oxo-N-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidine-3-carboxamide
2-butoxy-1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-(2-chloro-4-fluoro-5-methylphenyl)-3-(2-hydroxyethyl)-3-[(3-methylthiophen-2-yl)methyl]urea
1-benzyl-8-[(2-hydroxy-5-methoxyphenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 5-[(cyclohexylmethyl)amino]-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)amino]pyridine-3-carbonitrile
4-(4-ethyl-1H-pyrazol-5-yl)-1-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
(3S,4R)-4-methyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine-3,4-diol
(3aR,6aR)-2-[(2-chloro-4-fluorophenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3S,4R)-1-[(5-chloro-2-fluorophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(3R,4R)-1-[6-(3-fluorophenyl)pyridine-3-carbonyl]-4-(hydroxymethyl)piperidin-3-ol
3-[3-(5-methyl-1,2-oxazol-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
2-(4-fluorophenyl)-N-[1-(4-methyl-1H-imidazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
1-ethyl-8-(2-methylbutyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione