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4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]benzamide
1-amino-N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}cyclopropane-1-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[3-(3-methylphenyl)phenyl]piperidin-4-amine
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carboxamide
5-({cyclohexyl[2-(ethylsulfanyl)ethyl]amino}methyl)-2-methoxybenzoic acid
ethyl 4-[(3-fluorophenyl)methyl]-1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidine-4-carboxylate
(2S,4R)-1-[(4-methoxy-3-methylphenyl)methyl]-N,N-dimethyl-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
4-(1-benzoxepine-4-carbonyl)morpholine-2-carboxylic acid
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[(3,4-dimethoxyphenyl)methyl]-3-hydroxy-N-(1-methoxypropan-2-yl)benzamide
1-(6-chloro-2-methylpyridin-3-yl)-3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]urea
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-methyl-3-[3-(pyridin-4-yl)propyl]-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
9-methoxy-3-[(4-methoxyphenyl)methyl]-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
3-(2-amino-1H-1,3-benzodiazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
2-cyclohexyl-N-(pyridin-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
1-(carbamoylmethyl)-N-[(2,5-dimethoxyphenyl)methyl]piperidine-3-carboxamide
3-methoxy-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-(1,2-diphenylethyl)-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
(1R,3S)-3-(2-aminoethoxy)-7-[5-(methoxymethyl)thiophene-2-carbonyl]-7-azaspiro[3.5]nonan-1-ol
4-{[1-(pyrazin-2-yl)piperidin-4-yl]methyl}morpholine
2-[8-(2,3-dihydro-1-benzothiophene-2-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
2-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}-2H-chromene-3-carboxamide
[5-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)furan-2-yl]methanol
2-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)pyridine-3-carboxylic acid
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
1-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}piperidine-4-carboxamide
2-ethyl-8-(pent-2-yn-1-yl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 1-({4-[2-(dimethylamino)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
methyl[2-(morpholin-4-yl)propyl](pyridin-2-ylmethyl)amine
3-(5-{[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
3-phenyl-N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}-1H-pyrazole-5-carboxamide
7-fluoro-3-[({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amino)methyl]-1,2-dihydroquinolin-2-one
N-[2-(2-chlorophenyl)ethyl]-3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(2-methylpropyl)piperidin-3-yl]propanamide
4-(4-chlorophenyl)-N-[2-(pyrrolidin-1-yl)ethyl]butanamide
2-(4-ethylpiperazin-1-yl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
N-({8-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-fluorobenzamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-pyrazole-3-carboxamide
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-(2-methoxyethyl)-1-(3-methylbutyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-methoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
1-[(4aR,8aR)-6-(propane-2-sulfonyl)-decahydro-1,6-naphthyridin-1-yl]-4-(thiophen-2-yl)butan-1-one
2-[(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-8-methylquinolin-3-yl}methanol
7-(1,3-benzothiazol-2-yl)-9-methoxy-4-[(5-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-4-(4-methoxyphenyl)butane-1,4-dione
1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one