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3-{[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]methyl}benzoic acid
(2S,4S)-4-amino-N-ethyl-1-{2-[(4-methoxyphenyl)amino]-2-methylpropanoyl}pyrrolidine-2-carboxamide
N-{1-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-methoxyacetamide
N-(cyclopropylmethyl)-5-(2-methoxyacetamido)-N-(oxolan-2-ylmethyl)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(6-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-{[1-(3,4-dimethylbenzoyl)piperidin-3-yl]methyl}-4-fluorobenzamide
4-{2-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]propyl}-2-methoxyphenol
4-({4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)pyridin-2-ol
1-benzyl-8-[(3-hydroxyphenyl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-chloro-6-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperazin-1-yl}pyridazine
2-{3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}benzene-1,3-diol
2-(adamantan-1-yl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]acetamide
6-(1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
[1-({methyl[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}methyl)cyclopentyl]methanol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-5-methoxybenzamide
(3S,9aR)-8-(3-chlorobenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-(1-methyl-1H-pyrazol-3-yl)piperidine
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(2,6-difluoro-3-methylphenyl)-1-[2-(oxolan-3-yl)ethyl]-1H-imidazole
[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl](pyridin-2-yl)methanol
4-{3-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]propoxy}benzamide
N,6-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyridazin-3-amine
4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
9-[3-(4-fluorophenyl)propanoyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl](methyl)amino}-N-methylacetamide
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-[4-(propan-2-yl)piperazin-1-yl]pyridine-3-carboxamide
2-(3-hydroxyadamantan-1-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]acetamide
2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-N-cyclopentyl-2-oxoacetamide
[(2S,6S)-4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
5-[4-(azepane-1-carbonyl)-6,8-dimethylquinolin-2-yl]-N-methylpyrimidin-2-amine
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(1H-pyrazole-3-carbonyl)-1,4-diazepan-5-one
5-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
5-[(isoquinolin-5-yloxy)methyl]-N-[1-(4-methylphenyl)propyl]-1,2-oxazole-3-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(propan-2-yl)piperidine-3-carboxamide
5-[1-(4-acetylbenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
4-(2-fluorophenoxy)-1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
4-{1-[2-(4-chlorophenyl)ethyl]-6-oxopiperidine-3-carbonyl}-1-cyclohexylpiperazin-2-one
8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(2-hydroxyphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
1-{1-[2-(methylcarbamoyl)ethyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-methyl-4-({4-methyl-5-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
3-(furan-2-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-methoxy-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 1-[7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carbonyl]piperidine-3-carboxylate