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6-(benzyloxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(1,2,5-thiadiazole-3-carbonyl)-1,4-diazepan-2-one
[4-benzyl-1-(2,4-dimethylbenzoyl)piperidin-4-yl]methanol
N-{1-[1-(3-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
3-{[butyl(furan-2-ylmethyl)amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
2-benzyl-5-formamido-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-1H-1,3-benzodiazole-7-carboxamide
1-{2-[1-(2,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}-5-methyl-1H-1,2,3,4-tetrazole
1-cyclohexyl-N-methyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
(3aR,5S,6S,7aS)-2-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-octahydro-1H-isoindole-5,6-diol
4-(1H-imidazol-1-ylmethyl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-4-ol
1-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1H-pyrazol-1-yl)propan-1-one
ethyl 4-({[6-methyl-2-oxo-1-(prop-2-en-1-yl)-1,2-dihydroquinolin-3-yl]methyl}amino)piperidine-1-carboxylate
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-3-(4-hydroxyphenyl)benzamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
N-ethyl-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidine-3-carboxamide
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-[3-(2-oxoimidazolidin-1-yl)benzoyl]-decahydro-1,6-naphthyridin-2-one
1-ethyl-6-{[3-(pyridin-4-yl)azetidin-1-yl]methyl}-1H-indole
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)[(2-methylpyridin-4-yl)methyl]amine
(2S,4S)-4-amino-N-ethyl-1-{2-[5-oxo-2-(thiophen-2-yl)cyclopent-1-en-1-yl]acetyl}pyrrolidine-2-carboxamide
3-{1-[2-(4-methoxyphenoxy)acetyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-[3-(aminomethyl)phenyl]-3-({1-[ethyl(methyl)amino]cyclohexyl}methyl)urea
5-{1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-4-yl}-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
2-[1-(cyclohexylmethyl)-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-{3-[4-(4-hydroxyphenyl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
2-amino-6-(indolizin-2-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
2-(4-methyl-1H-pyrazol-1-yl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-(2,6-difluorophenoxymethyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(4S,4aS,8aS)-1-{[4-(2-hydroxyethoxy)phenyl]methyl}-4-phenyl-decahydroquinolin-4-ol
4-{[9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-3-(1,2-oxazolidin-2-yl)propanamide
3-chloro-N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]benzene-1-sulfonamide
N-{[3-(cyclopentyloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]-1,3-thiazole-5-carboxamide
4-chloro-N,N-diethyl-3-{[(morpholin-2-ylmethyl)carbamoyl]amino}benzamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2,5-dimethyl-N-(oxolan-2-ylmethyl)furan-3-carboxamide
N-[2-ethyl-4-(quinolin-3-yl)phenyl]acetamide
methyl 3-{[(3,5-dimethoxyphenyl)formamido]methyl}-5-(2-phenylacetamido)benzoate
N-(2-methyl-1-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
methyl(thiophen-2-ylmethyl){[3-({1-[4-(trifluoromethyl)benzenesulfonyl]piperidin-4-yl}oxy)phenyl]methyl}amine
(furan-3-ylmethyl)(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amine
5-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}({[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl})amine
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(dimethylamino)benzamide
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-[({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amino)methyl]pyrrolidin-2-yl]methanol
3-ethyl-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-1H-indole-2-carboxamide
N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-(pyrazin-2-yl)propanamide
3-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}benzonitrile
2-methoxy-N-({8-[(3-methylthiophen-2-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[2-(oxan-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclohexyl-4-(2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazin-2-one