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1-(2,2-dimethylpropyl)-3-hydroxy-3-[({imidazo[1,2-a]pyridin-3-ylmethyl}amino)methyl]piperidin-2-one
N-[2-(4-fluorophenyl)ethyl]-1-methyl-6-oxo-N-(pyridin-3-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
(1R,5R)-3-(pyrazin-2-yl)-6-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-(3-fluorophenyl)-3-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
3,4,7-trimethyl-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-indole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(pyrrolidine-1-sulfonyl)piperidin-3-ol
N-[4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
1-[(3-chlorophenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-benzyl-3-(2-methoxyethyl)-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(4-ethoxyphenyl)methyl]-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl}ethan-1-ol
3,5-dimethyl-1-(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}azetidin-3-yl)-1H-pyrazole
4-[(4-fluorophenyl)methyl]-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(3-ethylphenyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-3,5,7-trimethyl-1H-indole-2-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}propanamide
1-[(4-chlorophenyl)methyl]-N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-(4-methoxybutyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazine
N-methyl-3-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
2-(3-ethylphenyl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid
2-(2-{[methyl({2-[(4-methylphenyl)sulfanyl]ethyl})amino]methyl}phenoxy)acetamide
1-(1H-indazol-6-yl)-4-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperazin-2-one
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-4-(1H-pyrazol-1-yl)-N-(pyridin-4-ylmethyl)benzamide
(2S,4R)-4-cyclopentaneamido-N,N-diethyl-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
1-(3-chloro-2-methylphenyl)-5-[2-(1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
2,3-dimethoxy-N-[2-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)propyl]benzamide
8-phenylmethanesulfonyl-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-methyl-2-(4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
(4aS,7aR)-1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(9aR)-8-[(2,4-dimethylphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{2-hydroxy-3-[2-methoxy-4-({[(2-methoxyphenyl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
N-[(2,5-dimethoxyphenyl)methyl]-3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
5-(2,4-difluorophenoxymethyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,2-oxazole-3-carboxamide
4-(3-chlorophenoxy)-1-(1,4-dioxane-2-carbonyl)piperidine
ethyl 4-[4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carbonyl]piperazine-1-carboxylate
N-[(3S,4R)-1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}spiro[2.5]octane-1-carboxamide
4-cyclobutaneamido-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}benzamide
methyl 2-chloro-4-({[2-(2-methylpropanesulfonyl)ethyl]carbamoyl}amino)benzoate
2-{1-[(2-methylphenyl)methyl]-4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(1H-indol-3-yl)ethyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-cyclopentyl-1-methyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-methoxy-N-{2-[7-(2-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
2-(2-chlorophenoxy)-1-(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)ethan-1-one
5-(4-methyl-1,4-diazepan-1-yl)-2-[(3-methylquinoxalin-2-yl)methyl]-2,3-dihydropyridazin-3-one
methyl 1-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-2-carboxylate
2-{1-methyl-4-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]piperazin-2-yl}ethan-1-ol
N,5-dimethyl-4-{[(6-methylpyridin-2-yl)methyl]amino}-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide