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N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)pyridine-3-carboxamide
N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-phenylcyclopropane-1-carboxamide
5-(2,6-dimethoxyphenyl)-3-[4-(2-fluorophenyl)piperazin-1-yl]-1,2,4-triazine
3-(oxolan-3-yl)-5-[4-(1H-1,2,4-triazol-3-yl)phenyl]-1,2,4-oxadiazole
(1S,6R)-3-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
4-(3-methylpyridin-4-yl)-N-(1,2,3-thiadiazol-5-yl)-1,4-diazepane-1-carboxamide
ethyl (4aR,6R,8aS)-2-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline-8a-carboxylate
4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-1-benzyl-6-(cyclopropylmethoxy)-1,4-diazepan-2-one
3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
1-(azepan-1-yl)-3-[1-(2-hydroxyethyl)-3-methyl-1H-1,2,4-triazol-5-yl]propan-1-one
(2S)-1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-methyl-2-(propan-2-yl)piperazine
(1S,5R)-3-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4R)-4-(4-fluorophenyl)-1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-methyl-1-[3-(1-phenyl-5-propyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
[(1-benzylpiperidin-4-yl)methyl](1H-imidazol-2-ylmethyl)methylamine
1-[1'-(2-hydroxy-5-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-[2-(8-methoxyquinolin-5-yl)phenyl]ethan-1-amine
1-(3-fluorophenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-1H-pyrazole
5-[(2-ethoxyphenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-{[8-(2-oxo-2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
2-[(4-chlorophenyl)methyl]-N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-1,3-benzoxazole-5-carboxamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-5-methyl-1,3-oxazole-4-carboxamide
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-methyl-1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
2-methyl-4-[3-(morpholin-4-yl)piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
methyl (2S)-2-[2-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H-imidazol-1-yl]-2-phenylacetate
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-methyl-N-(thiophen-3-ylmethyl)acetamide
(1-{5-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-yl)methanol
1-(2-methoxyethyl)-5-[(4-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-cyclopropyl-5-[1-(2-hydroxyethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
(4aR,8aS)-1-[2-(2-fluorophenyl)ethyl]-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}butan-1-one
2-[methyl(2-phenylethyl)amino]-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
4-(1H-pyrazol-1-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]butan-1-one
1-(cyclopent-1-ene-1-carbonyl)-3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidine
3-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
6-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-4-oxo-4H-pyran-2-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
1-[(2R,3R)-2-hydroxy-3-(thiomorpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-methoxyethan-1-one
1-{[3-(cyclopentyloxy)phenyl]methyl}-4,4-difluoropiperidine
2-[(3-chlorophenyl)methyl]-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1,3-benzoxazole-6-carboxamide
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}propanamide
1-(2-chlorobenzoyl)-3-(3-methoxybenzoyl)piperidine
(1S,5R)-6-(cyclopropylmethyl)-3-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(4-ethylpiperazin-1-yl)-3-(2-methoxy-4-{[methyl(2-phenylethyl)amino]methyl}phenoxy)propan-2-ol
4-(2-methoxyacetyl)-N-[3-(methylsulfamoyl)phenyl]-1,4-diazepane-1-carboxamide
(1S,4S)-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-(4-methoxy-2-methylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-({[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]amino}methyl)-6-fluoroquinolin-4-ol