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(2S)-2-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)-3-methylbutanamide
4-(5-methoxyfuran-2-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-methyl-5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-phenylpyrimidine
2,4-dimethyl-5-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,3-thiazole
1-methanesulfonyl-4-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1,4-diazepane
1-(2,3-dihydro-1H-inden-2-yl)-4-(1H-imidazol-4-ylmethyl)-1,4-diazepane
1-(4-methoxyphenyl)-5-[2-(2-methyl-1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
9-(2-ethylpyridine-4-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
methyl 5-cyano-2-methyl-6-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyridine-3-carboxylate
2,4-dichloro-3-{[2-(3-hydroxypropyl)piperidin-1-yl]methyl}phenol
2,6-difluoro-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]benzamide
1-[(4-chlorophenyl)methyl]-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[3-({[4-(ethylamino)pyrimidin-2-yl]amino}methyl)piperidin-1-yl]-2-methylpropan-1-one
N-benzyl-6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-(cyclohexylmethyl)-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
3-(2-hydroxyphenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
5-(cyclohex-1-en-1-ylmethyl)-3-cyclopropyl-1H-1,2,4-triazole
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1H-indole-2-carboxamide
5-(3,4-difluorophenoxymethyl)-N-methyl-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
N-methyl-2-propyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1,3-thiazole-4-carboxamide
4-(hydroxymethyl)-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]azepan-4-ol
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(methylsulfanyl)propan-1-one
2-amino-4-(4-hydroxy-3-methylphenyl)-6-(pyrimidin-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-1,5-dimethyl-1H-pyrazole-3-carboxamide
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-acetamidopropanamide
5,6-dimethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)pyridine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-ol
1-(2-methylpropyl)-8-[(3-phenoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[6-(dimethylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
(3R,5S)-N-[(dimethyl-1,3-thiazol-5-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(3,4-dimethoxyphenyl)acetamide
5-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4-(propan-2-yl)-1,2,3-thiadiazole
{4-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]phenyl}methanol
(1R,3S)-3-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)cyclopentan-1-amine
(1S,5R)-6-methyl-N-(naphthalen-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(4-ethylphenyl)methyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
1-methyl-N,N-bis(2-methylpropyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-{[1-(2-hydroxyethyl)piperidin-3-yl]methyl}-N-methyl-1H-pyrazole-4-carboxamide
6-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine-1-sulfonamide
2-(2-chlorophenyl)-N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-[2-(1H-imidazol-2-yl)benzoyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(methylsulfanyl)propanamide
(2S,4S)-4-amino-N,N-diethyl-1-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)pyrrolidine-2-carboxamide
3-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propanamide
N-(oxolan-2-ylmethyl)-N-{[4-(thiophen-2-ylmethoxy)phenyl]methyl}-2H-1,3-benzodioxole-5-carboxamide