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(1R,2S)-N-tert-butyl-2-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}cyclohexane-1-carboxamide
3-{[(4-methylphenyl)methyl]amino}-N-[(1S)-1-phenylethyl]-5-[(propan-2-yl)sulfamoyl]benzamide
6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one
N,2-diethyl-4-methyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-1,3-oxazole-5-carboxamide
2-[(1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
5-methoxy-1,2-dimethyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-indole-3-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-(6-fluoro-4-methylquinazolin-2-yl)piperidine-4-carboxamide
2,4-dimethyl-5-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,3-thiazole
2-methyl-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]propan-2-amine
1-(2,3-dihydro-1H-inden-2-yl)-4-(furan-2-carbonyl)-1,4-diazepan-6-ol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
2-(4-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperazin-1-yl)ethan-1-ol
(3R,9aR)-3-(2-methylpropyl)-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(1-butyl-1H-imidazol-2-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine
4-(hydroxymethyl)-3-[(2-phenylphenyl)methyl]-1,3-oxazolidin-2-one
2-({8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)benzonitrile
3-methyl-1-(propan-2-yl)-4-[3-(pyridin-2-ylmethoxy)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[2-(morpholin-4-ylmethyl)phenyl]-6-(2-phenylethyl)-3,4-dihydropyrimidin-4-one
N-[1-methyl-5-(2-methylpiperidine-1-carbonyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazol-7-yl]cyclobutanecarboxamide
4-{[6-(2,6-dimethoxyphenyl)pyridin-3-yl]methyl}morpholine
N-[(3R,4S)-4-cyclopropyl-1-[(3,5-difluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl]-3-hydroxypropanamide
N-[(3-methylpyridin-4-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-1-cyclopropyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
5-methoxy-3-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-indole-2-carboxamide
1-(azepan-1-yl)-3-[2-(azetidin-1-ylmethyl)-4-chlorophenoxy]propan-2-ol
3-{[(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
4,6-dimethyl-3-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,2-dihydropyridin-2-one
N-[(3-methyl-7-{2-[3-(trifluoromethyl)phenyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(piperidin-1-yl)acetamide
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-[methyl(propan-2-yl)amino]propan-1-one
4-hydroxy-2-(phenoxymethyl)-N-[1-(1,3-thiazol-2-yl)propyl]pyrimidine-5-carboxamide
N-methyl-3-[2-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]carbamoyl}amino)phenyl]propanamide
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-N-[(2-methoxyphenyl)methyl]propanamide
9-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-(1-cyclopentyl-3-oxopiperazin-2-yl)acetamide
2-cyclopentyl-N-(quinolin-2-ylmethyl)acetamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(pyridin-3-yl)ethyl]propanamide
6-(2,5-dimethylfuran-3-yl)-N-ethyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
7-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N3-(4-methylpyrimidin-2-yl)-N1-(pyridin-3-yl)propane-1,3-diamine
4-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyrimidin-2-amine
4-(2-methoxyphenoxy)-1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
3-{2-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-(1H-1,2,3-benzotriazole-5-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-7-ethyl-2,7-diazaspiro[4.5]decan-6-one
2-methyl-6-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
methyl 6-{[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyridine-2-carboxylate
N-{2-[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
(furan-3-ylmethyl)(methyl){[3-({1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopentanecarboxamide