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N-[2-(4-fluorophenyl)ethyl]-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxylic acid
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(pyridin-3-yloxy)propyl]amine
1-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)azepan-2-one
5-fluoro-2-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane-6-carbonyl)-1H-indole
N-cyclopropyl-3-{1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-4-yl}propanamide
methyl 1-ethyl-5-[(3-hydroxy-3-methylbutan-2-yl)amino]-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-amino-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]pyridine-2-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(2-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
6-methyl-3-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-cyclopropyl-9-[2-hydroxy-2-(4-methoxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 5-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(2-amino-1,3-benzothiazole-5-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-(oxolan-2-ylmethyl)-N-(3-phenylprop-2-yn-1-yl)pyrazine-2-carboxamide
methyl 9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-3-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-(4-methylpiperazin-1-yl)ethan-1-one
N,N-dimethyl-5-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)isoquinoline-5-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(oxolan-2-ylmethyl)-N-propylbenzamide
2-[3-(2-methylpropyl)-5-[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]-1H-1,2,4-triazol-1-yl]pyridine
(2S,4S,5R)-5-(4-chlorophenyl)-4-(cyclobutylcarbamoyl)-1,2-dimethylpyrrolidine-2-carboxylic acid
8-methoxy-2-methyl-4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-(cyclohexylsulfamoyl)-N-(2,3-dihydro-1H-inden-2-yl)-5-(1H-pyrazol-3-yl)benzamide
N-[(3R,5S)-5-({[(2-methylphenyl)carbamoyl]methyl}carbamoyl)pyrrolidin-3-yl]thiophene-2-carboxamide
5-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-4-methyl-1H-imidazole
N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]furan-2-carboxamide
2,3-dimethyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}quinoxaline-6-carboxamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-methoxyethan-1-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyridin-4-yl)propanamide
1-(3-methylbutyl)-4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-pyrazole
1-[(3,4-dimethylphenyl)methyl]-4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazin-2-one
2-[(4-chlorophenyl)methyl]-N-[2-(1,3-thiazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
methyl 3-benzamido-5-{[2-(3-methyl-1H-pyrazol-1-yl)acetamido]methyl}benzoate
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethylpyrimidine-5-carboxamide
2-[(6-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-yl)amino]ethan-1-ol
N-(3,3-diphenylpropyl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-3-propylmorpholine
N-[(1S,2R)-2-[(1-benzylpiperidin-4-yl)amino]cyclobutyl]-2-(methylsulfanyl)acetamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(thiophen-2-ylmethyl)piperazine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(2-methoxy-5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methanol
1-{1-[3-(3-methylphenyl)phenyl]piperidin-4-yl}piperidine-4-carbonitrile
1-[(2,3-difluorophenyl)methyl]-3-({[2-(dimethylamino)ethyl]amino}methyl)-3-hydroxypiperidin-2-one