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1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
1-(3-methylpyridin-2-yl)-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazine
(3aS,6aS)-2-cyclopropanecarbonyl-5-(5-methyl-1,3-oxazole-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[2-(methylsulfamoyl)ethyl]sulfamoyl}-N-(propan-2-yl)benzamide
1,8-dibenzyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-6-methylpyridine-2-carboxamide
3-methyl-8-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(3-methylpyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{1-[(3-carboxy-4-methoxyphenyl)methyl]piperidin-4-yl}piperidine-4-carboxylic acid
4-oxo-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydroquinazoline-2-carboxamide
5-(1-methyl-1H-1,3-benzodiazol-2-yl)-N-propylpyrimidin-2-amine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[6-(1-hydroxyethyl)pyridin-2-yl]piperidine-4-carboxylic acid
N-methyl-1-{2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(thiophen-2-ylmethyl)piperidine-4-carboxamide
N-(1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
2-(3-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-3-oxopropyl)-2,3-dihydro-1H-isoindol-1-one
(3S,4S)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3,4-diol
(3R,4S)-1-(2-methoxybenzenesulfonyl)-4-(propan-2-yl)pyrrolidin-3-amine
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
(1S,5R)-6-benzyl-3-[2-(3-methoxyphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-4-[3-(thiophen-2-yl)propanoyl]-1,4-diazepan-2-one
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-{spiro[2.5]octan-1-ylmethyl}propanamide
N-[2-(4-chlorophenyl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
4-{5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}morpholine
3-{1-[4-(2-methoxyphenyl)benzoyl]piperidin-3-yl}propanamide
N-methyl-5-(oxolan-2-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}thiophene-2-carboxamide
5-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}-2-methoxybenzoic acid
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-4-(trifluoromethyl)benzamide
(5S,9aS,9bS)-5-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)-5,6-dihydro-1,4-dioxine-2-carboxamide
[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-(naphthalen-2-yl)acetamide
3-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-4,5,6-trimethyl-1,2-dihydropyridin-2-one
N-(1-hydroxypropan-2-yl)-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
3-{imidazo[1,2-a]pyridin-2-yl}-5-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazole
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-(oxolan-3-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-[4-(cyclohexylmethyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
11-{[(3-fluorophenyl)methyl]amino}-4-[2-(pyridin-2-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-[(3-fluorophenyl)methyl]-5-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-3-(2-methylpropyl)imidazolidine-2,4-dione
1-(3-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-(1-methylcyclopropyl)propan-1-one
1-(2-ethylpyrimidine-5-carbonyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
benzyl({[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})ethylamine
dimethyl[2-(2-{1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
methyl 4-{4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}benzoate
3,5-dimethyl-1-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]-1H-pyrazole
4-(1-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine