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N-[(2R,3R)-2-methoxy-1'-(5-propyl-1,2-oxazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}({[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl})amine
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
(2E)-N-{[5-chloro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(4-methoxyphenyl)prop-2-enamide
1-[(4-methanesulfonylphenyl)methyl]-4-(3-methylphenoxy)piperidine
N-({3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-(2-methyl-1H-indol-3-yl)acetamide
2-(1,2-benzoxazol-3-yl)-1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}ethan-1-one
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methoxyphenol
2-(morpholin-3-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]ethan-1-one
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-[(6-methylpyridin-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(1R,5R)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-(3,5-dimethylphenyl)-3-(4-methoxy-2-methylbenzoyl)piperidine-1-carboxamide
3-methyl-2-oxo-N-(1-phenyl-1H-pyrazol-5-yl)-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[1-(6-methoxynaphthalen-2-yl)ethyl]pyrrolidin-2-one
1-{2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-oxoethyl}piperidin-2-one
N-[3-(propan-2-yloxy)propyl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
ethyl 1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidine-4-carboxylate
3,4-dimethyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-5-sulfamoylbenzamide
2-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-benzyl-N-(1H-indol-4-ylmethyl)-1,3-benzoxazole-5-carboxamide
2-[2-(1,4-oxazepan-4-ylmethyl)phenyl]-6-propyl-3,4-dihydropyrimidin-4-one
1-ethyl-2-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,2-dihydropyridine-4-carboxamide
ethyl 4-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-amido}piperidine-1-carboxylate
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-methyl-N-(oxolan-3-yl)-1H-pyrazole-4-carboxamide
ethyl 4-oxo-5-phenoxy-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxylate
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
3-{1-[(3,7-dimethyl-1H-indol-2-yl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-(2-fluorophenyl)-3-(1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)propanamide
(3R,4R)-1-(4-ethyl-5-methylpyrimidin-2-yl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(1,3-thiazol-4-yl)ethyl]piperidin-2-one
1-(5-tert-butyl-1H-1,3-benzodiazol-2-yl)ethane-1,2-diol
6-(4-methyl-3-oxopiperazin-1-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-phenyl-1H-pyrazole
2-{[(3R,5S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]sulfanyl}-4,6-dimethylpyrimidine
3,5-difluoro-N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
1-(morpholin-4-yl)-3-[2-(pyridin-3-yl)phenoxy]propan-2-ol
2-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetamide
1-cyclobutanecarbonyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]piperidine-4-carboxamide
5-[(4-fluorophenyl)methyl]-5-{3-[3-(2-methylphenyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
methyl 5-[2-(ethanesulfonyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-(6-chloro-2H-1,3-benzodioxol-5-yl)-3-cyclobutyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
6-(2-aminoethyl)-N,2-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
N-({7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzenesulfonamide
3-{2-oxo-2-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethyl}-1,3-oxazolidin-2-one
2-methyl-4-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1,3-thiazole
2-[(3,4-difluorophenyl)methyl]-8-(morpholine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one