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1-(4-methylpiperazin-1-yl)-3-[5-(pyridin-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propan-1-one
N-({8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
(2S)-2-amino-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
1-{2-[(4-ethylpiperazin-1-yl)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-phenyl-4-{[2-(propylamino)pyrimidin-5-yl]methyl}piperazin-2-one
2-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
2,6-dimethyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}quinoline-4-carboxamide
(3aS,7aR)-5-methyl-2-[1-(2-phenylethyl)piperidin-4-yl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-cycloheptyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
(2S)-2-{2-[(2-ethoxyphenyl)carbamoyl]acetamido}-3-methylbutanoic acid
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[4-(morpholin-4-yl)butyl]amine
2-{4-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-3-methyl-2-oxopiperazin-1-yl}acetic acid
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6-(morpholine-4-carbonyl)pyrazin-2-amine
1-cyclopropyl-4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
2-chloro-5-acetamido-N-[(3S,4R)-4-ethoxyoxolan-3-yl]benzamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
6-(2-chlorophenyl)-N-cyclobutyl-7-(cyclopropylmethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
8-[(4-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-5-hydroxy-1,2-dimethyl-1H-indole-3-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(5-methylthiophene-2-carbonyl)pyrrolidin-3-yl]methanol
1-{[2-(trifluoromethoxy)phenyl]methyl}piperidine-2,6-dione
2-amino-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-6-hydroxy-5H-indeno[1,2-b]pyridine-3-carbonitrile
1-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
4-[(2-chloro-4,6-dimethoxyphenyl)methyl]-1-cyclopentylpiperazin-2-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
[(1-benzyl-1H-imidazol-2-yl)methyl](methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
[4-(4-phenoxyphenyl)pyridin-2-yl]methanol
(3S,4R)-1-(8-chloro-2-methylquinoline-4-carbonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
6-[(2-chlorophenyl)methyl]-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{[1-(1H-indol-2-ylmethyl)pyrrolidin-3-yl]methyl}-3-methylpyridine-4-carboxamide
N-[(3-chlorophenyl)methyl]-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3,6,7-trimethyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1-benzofuran-2-carboxamide
4-({4-[(3S)-3-ethylmorpholine-4-carbonyl]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
6-[3-(3,4-diethoxyphenyl)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(3-ethoxypropyl)amine
1-(6-chloro-1,3-benzothiazol-2-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
4,6-dimethyl-2-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,2-dihydropyridine-3-carboxamide
(3S,4R)-1-(isoquinoline-5-carbonyl)-3-methoxypiperidin-4-amine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(methanesulfonylmethyl)-3-(2-methylpropyl)-1H-1,2,4-triazole
N-[2-(2,3-dimethoxyphenyl)ethyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
4-(1,3-diphenyl-1H-pyrazol-4-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2S,4R)-1-{[3-(2-methylphenyl)phenyl]methyl}-N-(2-methylpropyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-(6-chloro-2-methylpyridin-3-yl)-3-methyl-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]urea
N4-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-[(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
4-[3-(1H-pyrazol-1-yl)phenyl]-1-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazole
3,5-dichloro-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-methylbenzamide
N-[1-(7-{[5-(4-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]acetamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(pentan-3-yl)piperidin-4-ol