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[(3R,4R)-1-(3-phenylbenzoyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
6-methoxy-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
7-fluoro-2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-methylquinoline
N-(pyrazin-2-yl)-2-{[1-(thiophen-2-yl)propan-2-yl]amino}acetamide
3-{1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}-N-cyclopropylpropanamide
N-methyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(1,3-thiazol-2-ylmethyl)acetamide
2-(2-chloro-4-fluorophenoxymethyl)-4-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1,3-oxazole
1-{[(2-cyclopentyl-2-phenylethyl)carbamoyl]methyl}piperidine-4-carboxamide
4-[(2-methylphenyl)sulfanyl]-1-(oxolane-3-carbonyl)piperidine
3-{3-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]propyl}-1H-indole
N-[(2R,3R)-1'-[(2,3-dimethoxyphenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
4-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-N-(furan-2-ylmethyl)pyridine-2-carboxamide
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-(3-methoxypropyl)piperidine
2-{[3-(2-oxopyrrolidin-1-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(3-{[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
N-(3-chloro-4-methoxyphenyl)-6-[1-(morpholin-4-yl)cyclohexanecarbonyl]-6-azaspiro[2.5]octane-1-carboxamide
N-({7-[4-(4-fluorophenyl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
2-(methylsulfanyl)-5-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]pyrimidine
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-(piperidine-1-carbonyl)piperidine
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-6-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-3-methanesulfonylpropan-1-one
2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)-1-methyl-1H-1,3-benzodiazole
1-(4-{[4-(hydroxymethyl)-4-[(4-methoxyphenyl)methyl]piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-methyl-5-{3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3,5-dimethyl-1H-pyrrole-2-carboxamide
N2-(2H-1,3-benzodioxol-5-ylmethyl)-N4-ethylpyrimidine-2,4-diamine
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
2-(4-{2-azaspiro[4.4]nonan-2-ylmethyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
7-[2-(2-chlorophenoxy)acetyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(diethylcarbamoyl)methyl]-N-[5-(morpholin-4-yl)pentyl]-1H-1,2,3-triazole-4-carboxamide
N-(1-methoxybutan-2-yl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-(4-fluorophenyl)piperidin-4-amine
2-(2-methoxyethyl)-6-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-1,3-benzoxazole
1-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}imidazolidin-2-one
(3S)-4-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
2-[2-(2,4-difluorophenoxy)acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-(methoxymethyl)thiophene-2-carboxamide
7-(3,4-dihydronaphthalen-2-yl)-4-propyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-benzyl-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-(2,4-dimethoxy-3-methylphenyl)-4-[(2-ethyl-1H-imidazol-1-yl)methyl]-5-methyl-1,3-oxazole
methyl (2S,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(furan-2-amido)pyrrolidine-2-carboxylate
1-[4-(1,3-benzoxazole-2-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
4-[1-(3-phenylpropyl)-5-(5-propyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
1-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(1-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}piperidin-2-yl)ethan-1-ol
5-(morpholin-4-ylmethyl)-N-[1-(pyrimidin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-(3-methoxypropyl)acetamide