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4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)pyrimidine
(1R,5S)-3-[(8-chloroquinolin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{1-[(2-methoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
N-(3-cyclopentaneamidophenyl)-2-ethyl-2,5-dihydro-1H-pyrrole-1-carboxamide
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1H-1,3-benzodiazole
4-{[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}benzoic acid
3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}-2-(thiophen-3-ylmethyl)propan-1-ol
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
4-(hydroxymethyl)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]pyridine-2-carboxamide
ethyl 4-({4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazine-1-carboxylate
2-[methyl(piperidin-4-yl)amino]-N-{[1-(phenoxymethyl)cyclopropyl]methyl}acetamide
propan-2-yl (1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
1-[6-(4-ethylpiperazin-1-yl)pyridine-3-carbonyl]-4-phenylazepane
3-[2-(3-chlorophenyl)acetyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
{[(1R,5S,6S)-3-(2-methoxybenzenesulfonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
1-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}azetidin-3-ol
3-{2-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-{[(2S,4S)-4-fluoro-1-(2-methoxypyridine-3-carbonyl)pyrrolidin-2-yl]methyl}morpholine-4-carboxamide
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)methylamine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
5-methanesulfonyl-N-[(2-methoxyphenyl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
2-methoxy-1-(4-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
{2-[4-(5-fluoro-1H-indole-2-carbonyl)morpholin-2-yl]ethyl}dimethylamine
3-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-ol
(2S,4R)-4-amino-N-methyl-1-{2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}pyrrolidine-2-carboxamide
2-(pyridin-3-ylmethyl)-8-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(1-cyclobutylpiperidin-4-yl)oxy]-N-(2-phenylethyl)benzamide
N-[3-(pyrrolidin-1-yl)propyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(2R)-2-amino-N-[(4-ethylphenyl)methyl]-3-hydroxy-N-(2-methoxyethyl)propanamide
9-[(2S)-1-ethylpyrrolidine-2-carbonyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(5-{[2-(methylsulfanyl)phenyl]carbamoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
(2S)-N2-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrrolidine-1,2-dicarboxamide
1-{2-[4-(ethanesulfonyl)piperazin-1-yl]pyrimidin-4-yl}piperidin-3-ol
5-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-methyl-1H-1,3-benzodiazole
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
(1R,5R)-6-[2-(4-chlorophenoxy)ethyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
5-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[(2R,3R)-2-methoxy-1'-[3-(methylsulfanyl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
(4aR,7aS)-1-ethyl-4-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[2-(2-hydroxyethyl)-3-oxopiperazin-1-yl]methyl}-N-(5-methyl-1,3-thiazol-2-yl)benzamide
2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methylacetamide
1,6-dimethyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-({3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
4-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}benzene-1-sulfonamide
4-[(4-methoxy-3-methylphenyl)methyl]-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)piperazin-2-one
1-[(2-chlorophenyl)methyl]-3-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
3-cyclohexyl-N-(2-oxoazepan-3-yl)-1H-pyrazole-4-carboxamide
N-[(2-methyl-1H-imidazol-4-yl)methyl]-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopentanamine
N-[(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide