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3-(3,4-dimethoxybenzoyl)-1-(furan-2-carbonyl)piperidine
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
2-amino-N-[(5-methylpyrazin-2-yl)methyl]-4-phenylpyrimidine-5-carboxamide
[(3-{2-[4-(5-chloro-3-methyl-1H-indole-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(1,3-thiazol-4-ylmethyl)amine
2-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
N-[(3S,4R)-1-[2-(4-chloro-2-methylphenoxy)acetyl]-4-propylpyrrolidin-3-yl]acetamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[4-(methylsulfanyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrazin-2-amine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S)-4-{5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carbonyl}-1,3-dimethylpiperazin-2-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
N-[3-(morpholin-4-yl)propyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
ethyl 4-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
3-(4-methyl-1,3-thiazol-5-yl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}propanamide
(3R,4S)-4-{4-[(5-chlorofuran-2-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
(3R,4S)-4-[methyl({[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl})amino]oxolan-3-ol
(3R,9aR)-8-(3,5-difluorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
5-methyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(quinoline-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
1-(7-chloroquinolin-4-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
6-methyl-2-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)acetamide
2-cyclopropyl-9-(4-ethylbenzenesulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
(7S,9aR)-7-[(4-chlorophenyl)methyl]-N-cyclohexyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
methyl 9-(benzyloxy)-3-[(3-fluoro-4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{2-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
6,8-dimethyl-3-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}pyridine-4-carboxylic acid
1-benzyl-5-[(3,4-difluorophenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-hydroxy-2-methyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]pyrimidine-5-carboxamide
2-{4-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
{1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidin-2-yl}methanol
4-{3-[(2,2,6,6-tetramethylpiperidin-4-yl)amino]butyl}phenol
N-(1-{1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
2-[3-(2-methoxyethyl)-5-[1-(pyrrolidin-1-yl)propyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-{3-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,3S)-3-(2-hydroxyethoxy)-7-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
1-methyl-4-({5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)piperazine
1-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-4-ol
3-({[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-methyl-4-(2-methylphenyl)piperazine
N-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N,2,2,6,6-pentamethylpiperidin-4-amine
4-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]pyrimidine-5-carboxylic acid
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-(3-phenylpropyl)propanamide