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{[4-(difluoromethoxy)phenyl]methyl}({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl})(2-methoxyethyl)amine
[1-(1-benzothiophen-2-ylmethyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
(1-{2-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]ethyl}piperidin-4-yl)methanol
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2,7-dimethylquinoline-4-carboxamide
2,4-dimethyl-5-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}-1,3-thiazole
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]methylamine
[(3R,4R)-1-[(6-fluoroquinolin-2-yl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-(1-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)methanesulfonamide
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}propanamide
2-cyclohexyl-1-[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]ethan-1-one
1-[2-(1H-pyrazol-3-yl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1,3-diethyl-5-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}-6-methyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
6-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(4-fluorophenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]acetamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-indole-6-carboxamide
N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
6-{[methyl(oxan-4-yl)amino]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[4-({[(3-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
methyl 1-(2-methylpropyl)-5-[(2-methylpropyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N,2,8-trimethyl-N-(piperidin-3-ylmethyl)quinoline-4-carboxamide
N-[1-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)propan-2-yl]-4-propylbenzamide
N3-butyl-1-cyclohexyl-4-oxo-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
8-methyl-2-propyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(1-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)-2-methoxyacetamide
(1-{1-[(2E,4E)-5-(4-fluorophenyl)penta-2,4-dien-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
3-[(2S)-2-amino-3-phenylpropanamido]-4-chloro-N,N-diethylbenzamide
N-methyl-4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]-1,3-thiazol-2-amine
1-[3-methoxy-4-({3-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidine-4-carbonitrile
1-{6-methyl-5-[5-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
2-(4-ethylpiperazin-1-yl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
(2S,4S)-4-amino-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(azepane-1-sulfonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(3S,4R)-1-[4-methoxy-3-(methoxymethyl)benzoyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-(pyridin-3-ylmethyl)-4-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(3-{[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]methyl}phenoxy)acetic acid
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-(methoxymethyl)-N-(oxolan-2-ylmethyl)furan-2-carboxamide
1-cyclopentyl-4-({[(8-fluoro-4-hydroxyquinolin-2-yl)methyl](methyl)amino}methyl)pyrrolidin-2-one
4-{[6-hydroxy-4-(1,2,5-oxadiazole-3-carbonyl)-1,4-diazepan-1-yl]methyl}benzoic acid
N-(1-{1-[(8-fluoroquinolin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
4-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-5-methoxy-1H-indole
5-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
4-[4-(3-ethylpiperazine-1-carbonyl)phenyl]-2-methylbut-3-yn-2-ol
N-{[7-(adamantane-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-5-carboxamide
3-ethyl-N-({7-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-{[4-(propan-2-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione