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1-(2,3-dihydro-1H-inden-2-yl)-4-({[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}amino)pyrrolidin-2-one
N-methyl-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
2-(3,5-dimethylbenzenesulfonyl)-2,8-diazaspiro[4.5]decane
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
3-[(dimethylamino)methyl]-1-(4-methyl-5-phenylthiophene-2-carbonyl)pyrrolidin-3-ol
N-[(2,3-dimethoxyphenyl)methyl]-2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetamide
4-[(2-fluorophenyl)methyl]-1-[3-(5-methylfuran-2-yl)butyl]-1,4-diazepan-5-one
7-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-1,3-diazepane-2,4-dione
1'-[6-(hydroxymethyl)pyridine-2-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)propanamide
5-(2-chlorophenyl)-2-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]furan-3-carboxamide
9-[(2S)-2-hydroxy-2-phenylacetyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(3-methoxypropyl)-6-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-{2-[1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
ethyl (1R,2S)-2-(4-phenyl-1H-imidazol-5-yl)cyclopropane-1-carboxylate
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
2-(3-methoxypropyl)-9-[(2-methylpyrimidin-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
9-oxo-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
2-(cyclohex-1-en-1-yl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-cyclohexyl-N-(prop-2-yn-1-yl)propanamide
2-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-2-yl}pyridine
1-[(2-chlorophenyl)methyl]-N-[(1-cyclopentylpiperidin-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(2,3-dimethylphenyl)-6-(4-methylpiperazine-1-carbonyl)pyrazine
2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
(4-benzyl-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-4-yl)methanol
2-(2-{1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
(2E)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(4-methoxyphenyl)prop-2-enamide
1-(1-methyl-1H-indole-6-carbonyl)-4-phenylpiperidine-4-carbonitrile
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-4-(piperidin-1-ylmethyl)benzamide
5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyrazin-2-ol
3-(3-methoxyphenyl)-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1-phenyl-1H-pyrazole
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]{[(1R,5S,6R)-3-(morpholine-4-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}amine
N-[(1R,3R)-3-aminocyclopentyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1,4-dimethyl 2-[3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamido]butanedioate
3-{1-[4-(2-phenylethyl)-1H-1,2,3-triazol-1-yl]propyl}pyridine
1-(2,3-dihydro-1-benzofuran-7-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
N-[(3S,4R)-1-(1-benzylpiperidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-[(dimethylamino)methyl]-1-(1,3,7-trimethyl-1H-indole-2-carbonyl)piperidin-3-ol
2,4-dimethoxy-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
5-cyclopropyl-3-(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)-1,2,4-oxadiazole
N,1,3-trimethyl-N-[(3-methylpyridin-4-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2H-1,3-benzodioxol-5-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidin-4-amine
N-({8-[2-(3-chlorophenoxy)propanoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-fluorobenzamide
N-(1-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
2,3-difluoro-6-methoxy-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]benzamide
2-methanesulfonyl-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)acetamide
N-[4-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]acetamide