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9-[3-(1H-pyrazol-1-yl)propanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 8-[2-(2-chlorophenoxy)acetyl]-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-methyl-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-cyclopropyl-2-(2-{[ethyl(pentan-2-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(3R,9aR)-3-benzyl-8-(4-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{3-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}azepan-2-one
3-(furan-2-yl)-N-methyl-3-phenyl-N-(prop-2-en-1-yl)propanamide
3-(4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
3-[1-(1-acetylpiperidin-4-yl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
6-cyclopentyl-1-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-{[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}-4-methylbenzoic acid
[3-(3-methoxypropyl)-1-(2-phenylethyl)piperidin-3-yl]methanol
[(3R,4R)-1-(2,6-dimethylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1-(3-phenylpropyl)piperidin-2-one
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
methyl 5-[2-(3,4-dichlorophenyl)morpholin-4-yl]pentanoate
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
6-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-2-methylheptan-2-ol
5-[1-(5-chloro-2-fluorobenzoyl)piperidin-4-yl]-3-(furan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N,2-dimethyl-5-phenyl-N-(1H-pyrazol-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(2S,4R)-N,N-diethyl-1-(4-fluorobenzoyl)-4-(2-methoxyacetamido)pyrrolidine-2-carboxamide
(4aR,7aS)-1-propanoyl-4-(quinoxaline-6-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,3S)-7-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-7-azaspiro[3.5]nonane-1,3-diol
6-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-3-phenylpyrazolo[1,5-a]pyrimidine
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)furan-3-carboxamide
4-(1H-indazole-3-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
N-{1-[(4-fluorophenyl)methyl]-5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-7-yl}acetamide
methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl][(1-propyl-1H-imidazol-2-yl)methyl]amine
7-(1-benzothiophen-3-yl)-4-(1-methyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[2-(4-methoxy-2-methylphenyl)pyridine-4-carbonyl]morpholine
8-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}-2-(morpholin-4-yl)quinoline
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1'-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]spiro[indene-1,4'-piperidine]
1-(1H-pyrazole-3-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
1-[3-(2-methylphenyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
(1-methyl-4-{[3-(3-methylbutoxy)phenyl]methyl}piperazin-2-yl)methanol
1-(1-methyl-1H-pyrazol-4-yl)-3-[3-(propan-2-yloxy)propyl]urea
5-(2,3-dichlorophenyl)pyridin-3-amine
2-(1,3-benzoxazol-2-yl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-2-[5-oxo-3-phenyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)benzamide
1-(4-{2-[9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
(2-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
5-(2,6-dimethylphenoxymethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
2,6-diamino-4-(2,1,3-benzothiadiazol-5-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-benzyl-1-cyclopropyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[2-(1H-pyrazol-4-yl)ethyl]quinoxaline-2-carboxamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,6-dimethyl-2-oxo-1,2-dihydropyridine-4-carboxamide