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9-(5-propylpyrimidin-4-yl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[4-(1H-pyrazol-5-yl)phenyl]pyrimidin-4-yl}piperidin-4-ol
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2-methoxypyridine
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-3-methylbut-2-en-1-one
N-benzyl-6-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(morpholin-2-yl)-N-{2-[3-(propan-2-yloxy)phenyl]ethyl}acetamide
N3-[(5-fluoro-2-methylphenyl)methyl]-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-1-(3-phenyl-1,2-oxazole-5-carbonyl)-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
5-methoxy-1-methyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-indole-2-carboxamide
6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-2-one
N-{1-[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
(2S,4S)-4-amino-1-{3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl}pyrrolidine-2-carboxylic acid
N-[(2R,3R)-2-methoxy-1'-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-pentanamidobenzamide
(butan-2-yl)[3-(1H-indazol-1-yl)propyl]amine
4-methyl-1-{2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
1-methyl-2-oxo-3-phenyl-N-propyl-1,8-diazaspiro[4.5]decane-8-carboxamide
3-(3-fluorophenyl)-4-{1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carbonyl}piperazin-2-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-[4-(methylsulfanyl)phenyl]acetamide
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-{[1-(pyridin-3-yl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-(3-fluorophenyl)-N-methyl-N-[(4-methylphenyl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[benzyl({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl})amino]butan-1-ol
1-[(4-methylphenyl)methyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
(4aR,8aS)-6-(2H-1,3-benzodioxol-5-ylmethyl)-1-(3,3-diphenylpropyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(azepan-1-yl)ethyl]-N,1-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-phenyl-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]pentan-1-one
1-{[4-(2-ethylpiperidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}-4-(2-fluorophenyl)piperazine
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-({1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}amino)-6-methylpyridine-3-carbonitrile
(1S,5R)-3-(5-cyclopropyl-1H-pyrazole-3-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-3-(1-methylpiperidin-2-yl)propan-1-one
methyl (2S)-3-(1H-indol-3-yl)-2-({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)propanoate
5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-4-yl)pyrimidine
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
N-(3-methoxypropyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
(3aR,6aR)-2-(2-methoxyethyl)-5-[4-(methylamino)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1H-1,3-benzodiazole-7-carboxamide
1-{4-[(3R,4S)-3-(dimethylamino)-4-(3-methoxyphenyl)pyrrolidin-1-yl]piperidin-1-yl}ethan-1-one
N-(1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
1-cyclopropyl-5-oxo-N-[3-(phenylsulfanyl)propyl]pyrrolidine-3-carboxamide
N-{[7-(2,5-dimethylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-2-carboxamide
2-methoxy-N-(1-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
benzyl({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl})ethylamine
3-[(2,2-dimethylpiperazin-1-yl)methyl]-N-[4-(2-hydroxyethyl)phenyl]benzamide
N,N-diethyl-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[3-(1H-imidazol-1-yl)propyl]benzamide
4-{[2-(methylsulfanyl)phenyl]methyl}piperazine-1-sulfonamide